BIX02189 (BIX 02189) supplier|cas# 1094614-85-3 |DC Chemicals|Supplier|Price|Buy
BIX02189 (BIX 02189) supplier|cas# 1094614-85-3 |DC Chemicals|Supplier|Price|Buy
DC Chemicals Supply: BIX02189 (BIX 02189) supplier,cas# 1094614-85-3, Cat No. DC5003, In stock
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Product name: BIX02189 (BIX 02189), Synonym: BIX 02189,BIX02189, Cat No. DC5003, Cas: 1094614-85-3, Chemical Name:(Z)-3-(((3-((dimethylamino)methyl)phenyl)amino)(phenyl)methylene)-N,N-dimethyl-2-oxoindoline-6-carboxamide, Molecular Formula: C27H28N4O2, MW: 440.54
BIX02189 (BIX 02189),cas 1094614-85-3, Purity: >98%. Best Price and quality in the market,DC Chemicals,Primary Manufacturer, confirmed by HNMR and HPLC. BIX02189 is a selective inhibitor of MEK5 with IC50 of 1.5 nM, also inhibits ERK5 catalytic activity with IC50 of 810 nM, and does not inhibit closely related kinases MEK1, MEK2, ERK2, and JNK2.
BIX 02189 is a selective MEK5/ERK5 inhibitor with an IC50 of 59 nM. BIX02189 was reported to inhibit catalytic function of purified, MEK5 enzyme.
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