FIIN2,FIIN-2|FGFR inhibitor|CAS 1633044-56-0|DC Chemicals
FIIN-2 is a potent, selective, irreversible and the next-generation covalent FGFR inhibitor.
Product name: FIIN-2 | Cat No. DC8330 |Cas: 1633044-56-0 |Other names: FIIN2,FIIN-2,FIIN 2 |Molecule formular: C35H38N8O4 |Molecule Weight: 634.3 |Purity>98%
FIIN-2 is a potent, selective, irreversible and the next-generation covalent FGFR inhibitor.
For research and scientific purpose only, not for human use.
2015年9月17日星期四
SLx-2119(KD-025) |Rock2 inhibitor|DC Chemicals
SLx-2119(KD-025) |Rock2 inhibitor|DC Chemicals
SLx-2119(KD-025) is a small molecule and selective inhibitor of ROCK2 with IC50 of 105 nM; > 200 fold selecivity over ROCK1(IC50 =24 uM)
Product name: SLx-2119(KD-025) | Cat No. DC8329 |Cas: 911417-87-3 |Other names: SLx2119(KD025)，SLx 2119(KD 025)，SLx2119，KD025 |Molecule formular: C26H24N6O2 |Molecule Weight: 452.51 |Purity>98%
SLx-2119(KD-025) is a small molecule and selective inhibitor of ROCK2 with IC50 of 105 nM; > 200 fold selecivity over ROCK1(IC50 =24 uM)
For research and scientific purpose only, not for human use.
SLx-2119(KD-025) is a small molecule and selective inhibitor of ROCK2 with IC50 of 105 nM; > 200 fold selecivity over ROCK1(IC50 =24 uM)
Product name: SLx-2119(KD-025) | Cat No. DC8329 |Cas: 911417-87-3 |Other names: SLx2119(KD025)，SLx 2119(KD 025)，SLx2119，KD025 |Molecule formular: C26H24N6O2 |Molecule Weight: 452.51 |Purity>98%
SLx-2119(KD-025) is a small molecule and selective inhibitor of ROCK2 with IC50 of 105 nM; > 200 fold selecivity over ROCK1(IC50 =24 uM)
For research and scientific purpose only, not for human use.
IRAK-1/4 Inhibitor|IL-1 kinases inhibitor|DC Chemicals
IRAK-1/4 Inhibitor|IL-1 kinases inhibitor|DC Chemicals
Interleukin-1 Receptor-Associated-Kinase-1/4 Inhibitor is a benzimidazole compound that acts as a cell-permeable, potent selective inhibitor of IL-1 kinases.
Product name: IRAK-1/4 Inhibitor | Cat No. DC8328 |Cas: 509093-47-4 |Other names: Interleukin-1 Receptor-Associated-Kinase-1/4 Inhibitor |Molecule formular: C20H21N5O4 |Molecule Weight: 395.42 |Purity>98%
Interleukin-1 Receptor-Associated-Kinase-1/4 Inhibitor is a benzimidazole compound that acts as a cell-permeable, potent selective inhibitor of IL-1 kinases.
For research and scientific purpose only, not for human use.
Interleukin-1 Receptor-Associated-Kinase-1/4 Inhibitor is a benzimidazole compound that acts as a cell-permeable, potent selective inhibitor of IL-1 kinases.
Product name: IRAK-1/4 Inhibitor | Cat No. DC8328 |Cas: 509093-47-4 |Other names: Interleukin-1 Receptor-Associated-Kinase-1/4 Inhibitor |Molecule formular: C20H21N5O4 |Molecule Weight: 395.42 |Purity>98%
Interleukin-1 Receptor-Associated-Kinase-1/4 Inhibitor is a benzimidazole compound that acts as a cell-permeable, potent selective inhibitor of IL-1 kinases.
For research and scientific purpose only, not for human use.
SANT-1|SANT1|Smo inhibitor|DC Chemicals
SANT-1|SANT1|Smo inhibitor|DC Chemicals
SANT-1 is a membrane permeable antagonist of the Shh (Sonic Hedgehog) signaling pathway by direct binding to Smo.
Product name: SANT-1 | Cat No. DC8327 |Cas: 304909-07-7 |Other names: SANT-1, SANT1,SANT 1 |Molecule formular: C23H27N5 |Molecule Weight: 373.49 |Purity>98%
SANT-1 is a membrane permeable antagonist of the Shh (Sonic Hedgehog) signaling pathway by direct binding to Smo.
For research and scientific purpose only, not for human use.
SANT-1 is a membrane permeable antagonist of the Shh (Sonic Hedgehog) signaling pathway by direct binding to Smo.
Product name: SANT-1 | Cat No. DC8327 |Cas: 304909-07-7 |Other names: SANT-1, SANT1,SANT 1 |Molecule formular: C23H27N5 |Molecule Weight: 373.49 |Purity>98%
SANT-1 is a membrane permeable antagonist of the Shh (Sonic Hedgehog) signaling pathway by direct binding to Smo.
For research and scientific purpose only, not for human use.
Kevetrin|activator of p53|DC Chemicals
Kevetrin|activator of p53|DC Chemicals
Kevetrin (thioureidobutyronitrile), is a water-soluble, small molecule and activator of the tumor suppressor protein p53, with potential antineoplastic activity.
Product name: Kevetrin HCl | Cat No. DC8326 |Cas: 66592-89-0 |Other names: |Molecule formular: C5H10ClN3S |Molecule Weight: 179.67 |Purity>98%
Kevetrin (thioureidobutyronitrile), is a water-soluble, small molecule and activator of the tumor suppressor protein p53, with potential antineoplastic activity.
For research and scientific purpose only, not for human use.
Kevetrin (thioureidobutyronitrile), is a water-soluble, small molecule and activator of the tumor suppressor protein p53, with potential antineoplastic activity.
Product name: Kevetrin HCl | Cat No. DC8326 |Cas: 66592-89-0 |Other names: |Molecule formular: C5H10ClN3S |Molecule Weight: 179.67 |Purity>98%
Kevetrin (thioureidobutyronitrile), is a water-soluble, small molecule and activator of the tumor suppressor protein p53, with potential antineoplastic activity.
For research and scientific purpose only, not for human use.
Ellipticine|DNA topoisomerase II inhibitor|DC Chemicals
Ellipticine|DNA topoisomerase II inhibitor|DC Chemicals
Ellipticine is a DNA intercalating agent and a DNA topoisomerase II inhibitor.
Product name: Ellipticine | Cat No. DC8325 |Cas: 519-23-3 |Other names: CCG-36483; CCG36483; CCG 36483; BRN-0221300; BRN0221300; BRN 0221300; DB-052047; K00071; LP00531; LS-133282; NSC 71795; NSC71795; NSC-71795; TCMDC-125546; VZ29809. elliptecine; ellipticine; Elliptisine |Molecule formular: C17H14N2 |Molecule Weight: 246.31 |Purity>98%
Ellipticine is a DNA intercalating agent and a DNA topoisomerase II inhibitor.
For research and scientific purpose only, not for human use.
Ellipticine is a DNA intercalating agent and a DNA topoisomerase II inhibitor.
Product name: Ellipticine | Cat No. DC8325 |Cas: 519-23-3 |Other names: CCG-36483; CCG36483; CCG 36483; BRN-0221300; BRN0221300; BRN 0221300; DB-052047; K00071; LP00531; LS-133282; NSC 71795; NSC71795; NSC-71795; TCMDC-125546; VZ29809. elliptecine; ellipticine; Elliptisine |Molecule formular: C17H14N2 |Molecule Weight: 246.31 |Purity>98%
Ellipticine is a DNA intercalating agent and a DNA topoisomerase II inhibitor.
For research and scientific purpose only, not for human use.
CCT244747|cas 1404095-34-6 |CHK1 inhibitor|DC Chemicals
CCT244747|cas 1404095-34-6 |CHK1 inhibitor|DC Chemicals
CCT244747 represents the first structural disclosure of a highly selective, orally active CHK1 inhibitor and warrants further evaluation alone or combined with genotoxic anticancer therapies.
Product name: CCT244747 | Cat No. DC8324 |Cas: 1404095-34-6 |Other names: CCT244747; CCT-244747; CCT 244747 |Molecule formular: C20H24N8O2 |Molecule Weight: 408.46 |Purity>98%
CCT244747 represents the first structural disclosure of a highly selective, orally active CHK1 inhibitor and warrants further evaluation alone or combined with genotoxic anticancer therapies.
For research and scientific purpose only, not for human use.
CCT244747 represents the first structural disclosure of a highly selective, orally active CHK1 inhibitor and warrants further evaluation alone or combined with genotoxic anticancer therapies.
Product name: CCT244747 | Cat No. DC8324 |Cas: 1404095-34-6 |Other names: CCT244747; CCT-244747; CCT 244747 |Molecule formular: C20H24N8O2 |Molecule Weight: 408.46 |Purity>98%
CCT244747 represents the first structural disclosure of a highly selective, orally active CHK1 inhibitor and warrants further evaluation alone or combined with genotoxic anticancer therapies.
For research and scientific purpose only, not for human use.
Eletriptan HBr |5-HT1B/1D receptor agonist|DC Chemicals
Eletriptan HBr |5-HT1B/1D receptor agonist|DC Chemicals
Eletriptan HBr is an orally active, selective 5-HT1B/1D receptor agonist.
Product name: Eletriptan HBr | Cat No. DC8323 |Cas: 177834-92-3 |Other names: Eletriptan hydrobromide |Molecule formular: C22H27BrN2O2S |Molecule Weight: 463.43 |Purity>98%
Eletriptan HBr is an orally active, selective 5-HT1B/1D receptor agonist.
For research and scientific purpose only, not for human use.
Eletriptan HBr is an orally active, selective 5-HT1B/1D receptor agonist.
Product name: Eletriptan HBr | Cat No. DC8323 |Cas: 177834-92-3 |Other names: Eletriptan hydrobromide |Molecule formular: C22H27BrN2O2S |Molecule Weight: 463.43 |Purity>98%
Eletriptan HBr is an orally active, selective 5-HT1B/1D receptor agonist.
For research and scientific purpose only, not for human use.
Anacardic acid|histone acetyltransferase inhibitor|DC Chemicals
Anacardic acid|histone acetyltransferase inhibitor|DC Chemicals
Anacardic acid inhibits the histone acetyltransferase (HAT) activity of the transcription co-activators p300 and p300/CREB-binding protein-associated factor (pCAF) with IC50 values of 8.5 and 5 µM, respectively.
Product name: Anacardic Acid | Cat No. DC8322 |Cas: 16611-84-0 |Other names: |Molecule formular: C22H36O3 |Molecule Weight: 348.52 |Purity>98%
Anacardic acid inhibits the histone acetyltransferase (HAT) activity of the transcription co-activators p300 and p300/CREB-binding protein-associated factor (pCAF) with IC50 values of 8.5 and 5 µM, respectively.
For research and scientific purpose only, not for human use.
Anacardic acid inhibits the histone acetyltransferase (HAT) activity of the transcription co-activators p300 and p300/CREB-binding protein-associated factor (pCAF) with IC50 values of 8.5 and 5 µM, respectively.
Product name: Anacardic Acid | Cat No. DC8322 |Cas: 16611-84-0 |Other names: |Molecule formular: C22H36O3 |Molecule Weight: 348.52 |Purity>98%
Anacardic acid inhibits the histone acetyltransferase (HAT) activity of the transcription co-activators p300 and p300/CREB-binding protein-associated factor (pCAF) with IC50 values of 8.5 and 5 µM, respectively.
For research and scientific purpose only, not for human use.
Entacapone|COMT inhibitor|DC Chemicals
Entacapone|COMT inhibitor|DC Chemicals
Entacapone is a specific, potent, peripherally acting catechol-O-methyltransferase (COMT) inhibitor with IC50 of 151 nM for PD treatment.
Product name: Entacapone | Cat No. DC8321 |Cas: 130929-57-6 |Other names: |Molecule formular: C14H15N3O5 |Molecule Weight: 305.29 |Purity>98%
Entacapone is a specific, potent, peripherally acting catechol-O-methyltransferase (COMT) inhibitor with IC50 of 151 nM for PD treatment.
For research and scientific purpose only, not for human use.
Entacapone is a specific, potent, peripherally acting catechol-O-methyltransferase (COMT) inhibitor with IC50 of 151 nM for PD treatment.
Product name: Entacapone | Cat No. DC8321 |Cas: 130929-57-6 |Other names: |Molecule formular: C14H15N3O5 |Molecule Weight: 305.29 |Purity>98%
Entacapone is a specific, potent, peripherally acting catechol-O-methyltransferase (COMT) inhibitor with IC50 of 151 nM for PD treatment.
For research and scientific purpose only, not for human use.
RVX-208|BET bromodomains inhibitor|DC Chemicals
RVX-208|BET bromodomains inhibitor|DC Chemicals
RVX-208(RVX 000222) is a small molecule that increases apolipoprotein A-I and high-density lipoprotein cholesterol in vitro and in vivo; is a BET bromodomain antagonist.
Product name: RVX-208 | Cat No. DC8320 |Cas: 1044870-39-4 |Other names: Apabetalone; RVX-000222; RVX208; RVX 208; RVX000222; RVX 000222 |Molecule formular: C20H22N2O5 |Molecule Weight: 370.4 |Purity>98%
RVX-208(RVX 000222) is a small molecule that increases apolipoprotein A-I and high-density lipoprotein cholesterol in vitro and in vivo; is a BET bromodomain antagonist.
RVX-208(RVX 000222) is a small molecule that increases apolipoprotein A-I and high-density lipoprotein cholesterol in vitro and in vivo; is a BET bromodomain antagonist.
Product name: RVX-208 | Cat No. DC8320 |Cas: 1044870-39-4 |Other names: Apabetalone; RVX-000222; RVX208; RVX 208; RVX000222; RVX 000222 |Molecule formular: C20H22N2O5 |Molecule Weight: 370.4 |Purity>98%
RVX-208(RVX 000222) is a small molecule that increases apolipoprotein A-I and high-density lipoprotein cholesterol in vitro and in vivo; is a BET bromodomain antagonist.
For research and scientific purpose only, not for human use.
Spautin 1|DUB inhibitor|DC Chemicals
Spautin 1|DUB inhibitor|DC Chemicals
Spautin 1 is an inhibitor of autophagy; inhibits USP10 and USP13 activity (IC50 values are 0.6 and 0.7 μM respectively) and promotes degradation of Vps34 (class III PI 3-kinase) complexes.
Product name: Spautin 1 | Cat No. DC8319 |Cas: 1262888-28-7 |Other names: Spautin-1,Spautin1 |Molecule formular: C15H11F2N3 |Molecule Weight: 271.26 |Purity>98%
Spautin 1 is an inhibitor of autophagy; inhibits USP10 and USP13 activity (IC50 values are 0.6 and 0.7 μM respectively) and promotes degradation of Vps34 (class III PI 3-kinase) complexes.
For research and scientific purpose only, not for human use.
Spautin 1 is an inhibitor of autophagy; inhibits USP10 and USP13 activity (IC50 values are 0.6 and 0.7 μM respectively) and promotes degradation of Vps34 (class III PI 3-kinase) complexes.
Product name: Spautin 1 | Cat No. DC8319 |Cas: 1262888-28-7 |Other names: Spautin-1,Spautin1 |Molecule formular: C15H11F2N3 |Molecule Weight: 271.26 |Purity>98%
Spautin 1 is an inhibitor of autophagy; inhibits USP10 and USP13 activity (IC50 values are 0.6 and 0.7 μM respectively) and promotes degradation of Vps34 (class III PI 3-kinase) complexes.
For research and scientific purpose only, not for human use.
ITE|Endogenous aryl hydrocarbon receptor (AhR) agonist|DC Chemicals
ITE|Endogenous aryl hydrocarbon receptor (AhR) agonist|DC Chemicals
ITE is an Endogenous aryl hydrocarbon receptor (AhR) agonist (Ki = 3 nM).
Product name: ITE | Cat No. DC8318 |Cas: 448906-42-1 |Other names: Aryl hydrocarbon receptor ligand |Molecule formular: C14H10N2O3S |Molecule Weight: 286.3 |Purity>98%
ITE is an Endogenous aryl hydrocarbon receptor (AhR) agonist (Ki = 3 nM).
For research and scientific purpose only, not for human use.
ITE is an Endogenous aryl hydrocarbon receptor (AhR) agonist (Ki = 3 nM).
Product name: ITE | Cat No. DC8318 |Cas: 448906-42-1 |Other names: Aryl hydrocarbon receptor ligand |Molecule formular: C14H10N2O3S |Molecule Weight: 286.3 |Purity>98%
ITE is an Endogenous aryl hydrocarbon receptor (AhR) agonist (Ki = 3 nM).
For research and scientific purpose only, not for human use.
GSK1324726A (I-BET726)|BET BRD inhibitor|DC Chemicals
GSK1324726A (I-BET726)|BET BRD inhibitor|DC Chemicals
GSK1324726A (I-BET726) is a novel, potent, and selective small molecule inhibitor of BET proteins with high affinity to BRD2 (IC50= 41 nM), BRD3 (IC50= 31 nM), and BRD4 (IC50= 22 nM).
Product name: GSK1324726A (I-BET726) | Cat No. DC8317 |Cas:
1300031-52-0 |Other names: GSK-1324726A,IBET726,GSK 1324726A,I BET726,I BET-726,I BET 726,I-BET-726 |Molecule formular: C25H23ClN2O3 |Molecule Weight: 434.91 |Purity>98%
GSK1324726A (I-BET726) is a novel, potent, and selective small molecule inhibitor of BET proteins with high affinity to BRD2 (IC50= 41 nM), BRD3 (IC50= 31 nM), and BRD4 (IC50= 22 nM).
For research and scientific purpose only, not for human use.
GSK1324726A (I-BET726) is a novel, potent, and selective small molecule inhibitor of BET proteins with high affinity to BRD2 (IC50= 41 nM), BRD3 (IC50= 31 nM), and BRD4 (IC50= 22 nM).
Product name: GSK1324726A (I-BET726) | Cat No. DC8317 |Cas:
1300031-52-0 |Other names: GSK-1324726A,IBET726,GSK 1324726A,I BET726,I BET-726,I BET 726,I-BET-726 |Molecule formular: C25H23ClN2O3 |Molecule Weight: 434.91 |Purity>98%
GSK1324726A (I-BET726) is a novel, potent, and selective small molecule inhibitor of BET proteins with high affinity to BRD2 (IC50= 41 nM), BRD3 (IC50= 31 nM), and BRD4 (IC50= 22 nM).
For research and scientific purpose only, not for human use.
SBI-0206965|autophagy kinase ULK1 inhibitor|DC Chemicals
SBI-0206965|autophagy kinase ULK1 inhibitor|DC Chemicals
SBI-0206965 is a potent, selective and cell permeable autophagy kinase ULK1 inhibitor.
Product name: SBI-0206965 | Cat No. DC8316 |Cas: N/A |Other names: SBI 0206965,SBI0206965 |Molecule formular: C21H21BrN4O5 |Molecule Weight: 489.33 |Purity>98%
SBI-0206965 is a potent, selective and cell permeable autophagy kinase ULK1 inhibitor.
For research and scientific purpose only, not for human use.
SBI-0206965 is a potent, selective and cell permeable autophagy kinase ULK1 inhibitor.
Product name: SBI-0206965 | Cat No. DC8316 |Cas: N/A |Other names: SBI 0206965,SBI0206965 |Molecule formular: C21H21BrN4O5 |Molecule Weight: 489.33 |Purity>98%
SBI-0206965 is a potent, selective and cell permeable autophagy kinase ULK1 inhibitor.
For research and scientific purpose only, not for human use.
Solcitinib（GLPG0778，GSK2586184）|DC Chemicals
Solcitinib（GLPG0778，GSK2586184）|DC Chemicals
Solcitinib, also known as GSK2586184 or GLPG0778, is a Janus kinase 1 (JAK1) inhibitor.
Product name: Solcitinib（GLPG0778，GSK2586184） | Cat No. DC8315 |Cas: 1206163-45-2 |Other names: GLPG 0778，GSK 2586184,GLPG-0778，GSK-2586184 |Molecule formular: C22H23N5O2 |Molecule Weight: 389.45 |Purity>98%
Solcitinib, also known as GSK2586184 or GLPG0778, is a Janus kinase 1 (JAK1) inhibitor.
For research and scientific purpose only, not for human use.
Solcitinib, also known as GSK2586184 or GLPG0778, is a Janus kinase 1 (JAK1) inhibitor.
Product name: Solcitinib（GLPG0778，GSK2586184） | Cat No. DC8315 |Cas: 1206163-45-2 |Other names: GLPG 0778，GSK 2586184,GLPG-0778，GSK-2586184 |Molecule formular: C22H23N5O2 |Molecule Weight: 389.45 |Purity>98%
Solcitinib, also known as GSK2586184 or GLPG0778, is a Janus kinase 1 (JAK1) inhibitor.
For research and scientific purpose only, not for human use.
Leuprolide Acetate|GnRH receptors agonist|DC Chemicals
Leuprolide Acetate|GnRH receptors agonist|DC Chemicals
Leuprolide acetate (Leuprorelin) is a GnRH analog; leuprolide acetate acts as an agonist at pituitary GnRH receptors.
Product name: Leuprolide Acetate | Cat No. DC8314 |Cas: 74381-53-6 |Other names: |Molecule formular: C61H88N16O14 |Molecule Weight: 1269.45 |Purity>98%
Leuprolide acetate (Leuprorelin) is a GnRH analog; leuprolide acetate acts as an agonist at pituitary GnRH receptors.
For research and scientific purpose only, not for human use.
Leuprolide acetate (Leuprorelin) is a GnRH analog; leuprolide acetate acts as an agonist at pituitary GnRH receptors.
Product name: Leuprolide Acetate | Cat No. DC8314 |Cas: 74381-53-6 |Other names: |Molecule formular: C61H88N16O14 |Molecule Weight: 1269.45 |Purity>98%
Leuprolide acetate (Leuprorelin) is a GnRH analog; leuprolide acetate acts as an agonist at pituitary GnRH receptors.
For research and scientific purpose only, not for human use.
BD-1047|σ receptors inhibitors|DC Chemicals
BD-1047|σ receptors inhibitors|DC Chemicals
BD 1047 dihydrobromide is a selective antagonist of σ receptors.
Product name: BD1047.2HBr | Cat No. DC8313 |Cas: 138356-21-5 |Other names: BD-1047，BD 1047 |Molecule formular: C13H20Cl2N2.2HBr |Molecule Weight: 437.04 |Purity>98%
BD 1047 dihydrobromide is a selective antagonist of σ receptors.
For research and scientific purpose only, not for human use.
BD 1047 dihydrobromide is a selective antagonist of σ receptors.
Product name: BD1047.2HBr | Cat No. DC8313 |Cas: 138356-21-5 |Other names: BD-1047，BD 1047 |Molecule formular: C13H20Cl2N2.2HBr |Molecule Weight: 437.04 |Purity>98%
BD 1047 dihydrobromide is a selective antagonist of σ receptors.
For research and scientific purpose only, not for human use.
NVP-231|ceramide kinase inhibitor|DC Chemicals
NVP-231|ceramide kinase inhibitor|DC Chemicals
NVP-231 is a potent, reversible inhibitor of ceramide kinase (IC50 = 12 nM).
Product name: NVP-231 | Cat No. DC8312 |Cas: 362003-83-6 |Other names: NVP-231,NVP 231，NVP231 |Molecule formular: C25H25N3O2S |Molecule Weight: 431.6 |Purity>98%
NVP-231 is a potent, reversible inhibitor of ceramide kinase (IC50 = 12 nM).
For research and scientific purpose only, not for human use.
NVP-231 is a potent, reversible inhibitor of ceramide kinase (IC50 = 12 nM).
Product name: NVP-231 | Cat No. DC8312 |Cas: 362003-83-6 |Other names: NVP-231,NVP 231，NVP231 |Molecule formular: C25H25N3O2S |Molecule Weight: 431.6 |Purity>98%
NVP-231 is a potent, reversible inhibitor of ceramide kinase (IC50 = 12 nM).
For research and scientific purpose only, not for human use.
Meleagrin|cas 71751-77-4|DC Chmeicals
Meleagrin|cas 71751-77-4|DC Chmeicals
Meleagrin is an antibiotic derived from a deep ocean, penicillin-producingP. chrysogenum.
Product name: Meleagrin | Cat No. DC8311 |Cas: 71751-77-4 |Other names: |Molecule formular: C23H23N5O4 |Molecule Weight: 433.5 |Purity>98%
Meleagrin is an antibiotic derived from a deep ocean, penicillin-producingP. chrysogenum.
For research and scientific purpose only, not for human use.
Meleagrin is an antibiotic derived from a deep ocean, penicillin-producingP. chrysogenum.
Product name: Meleagrin | Cat No. DC8311 |Cas: 71751-77-4 |Other names: |Molecule formular: C23H23N5O4 |Molecule Weight: 433.5 |Purity>98%
Meleagrin is an antibiotic derived from a deep ocean, penicillin-producingP. chrysogenum.
For research and scientific purpose only, not for human use.
BG-45|HDAC inhibitor|DC Chemicals
BG-45|HDAC inhibitor|DC Chemicals
BG45 is an HDAC class I inhibitor with selectivity for HDAC3 (IC50 = 289 nM). It inhibits HDAC1, HDAC2, and HDAC6 with greatly reduced potency (IC50s = 2, 2.2, and >20 µM, respectively).
Product name: BG-45 | Cat No. DC8310 |Cas: 926259-99-6 |Other names: BG45,BG 45 |Molecule formular: C11H10N4O |Molecule Weight: 214.2 |Purity>98%
BG45 is an HDAC class I inhibitor with selectivity for HDAC3 (IC50 = 289 nM). It inhibits HDAC1, HDAC2, and HDAC6 with greatly reduced potency (IC50s = 2, 2.2, and >20 µM, respectively).
For research and scientific purpose only, not for human use.
BG45 is an HDAC class I inhibitor with selectivity for HDAC3 (IC50 = 289 nM). It inhibits HDAC1, HDAC2, and HDAC6 with greatly reduced potency (IC50s = 2, 2.2, and >20 µM, respectively).
Product name: BG-45 | Cat No. DC8310 |Cas: 926259-99-6 |Other names: BG45,BG 45 |Molecule formular: C11H10N4O |Molecule Weight: 214.2 |Purity>98%
BG45 is an HDAC class I inhibitor with selectivity for HDAC3 (IC50 = 289 nM). It inhibits HDAC1, HDAC2, and HDAC6 with greatly reduced potency (IC50s = 2, 2.2, and >20 µM, respectively).
For research and scientific purpose only, not for human use.
Ruxolitinib Phosphate|DC Chemicals
Ruxolitinib Phosphate|DC Chemicals
Ruxolitinib Phosphate is a potent and selective Janus kinase (JAK1, IC50 = 5.9 nM and JAK2, IC50 = 5.7 nM) inhibitor.
Product name: Ruxolitinib Phosphate | Cat No. DC8309 |Cas: 1092939-17-7 |Other names: INCB018424,INCB-018424,INCB 018424 |Molecule formular: C17H18N6•H3O4P |Molecule Weight: 404.36 |Purity>98%
Ruxolitinib Phosphate is a potent and selective Janus kinase (JAK1, IC50 = 5.9 nM and JAK2, IC50 = 5.7 nM) inhibitor.
For research and scientific purpose only, not for human use.
Ruxolitinib Phosphate is a potent and selective Janus kinase (JAK1, IC50 = 5.9 nM and JAK2, IC50 = 5.7 nM) inhibitor.
Product name: Ruxolitinib Phosphate | Cat No. DC8309 |Cas: 1092939-17-7 |Other names: INCB018424,INCB-018424,INCB 018424 |Molecule formular: C17H18N6•H3O4P |Molecule Weight: 404.36 |Purity>98%
Ruxolitinib Phosphate is a potent and selective Janus kinase (JAK1, IC50 = 5.9 nM and JAK2, IC50 = 5.7 nM) inhibitor.
For research and scientific purpose only, not for human use.
SYM-2206|SYM2206|AMPA receptor inhibitor|DC Chemicals
SYM-2206|SYM2206|AMPA receptor inhibitor|DC Chemicals
SYM2206 is a novel, potent, non-competitive AMPA receptor antagonist (IC50 = 2.8 μM ).
Product name: SYM2206 | Cat No. DC8308 |Cas: 173952-44-8 |Other names: SYM2206,SYM 2206,SYM-2206 |Molecule formular: C20H22N4O3 |Molecule Weight: 366.42 |Purity>98%
SYM2206 is a novel, potent, non-competitive AMPA receptor antagonist (IC50 = 2.8 μM ).
For research and scientific purpose only, not for human use.
SYM2206 is a novel, potent, non-competitive AMPA receptor antagonist (IC50 = 2.8 μM ).
Product name: SYM2206 | Cat No. DC8308 |Cas: 173952-44-8 |Other names: SYM2206,SYM 2206,SYM-2206 |Molecule formular: C20H22N4O3 |Molecule Weight: 366.42 |Purity>98%
SYM2206 is a novel, potent, non-competitive AMPA receptor antagonist (IC50 = 2.8 μM ).
For research and scientific purpose only, not for human use.
QNZ-46|NMDA receptor inhibitor|DC Chemicals
QNZ-46|NMDA receptor inhibitor|DC Chemicals
QNZ is a NR2C/NR2D-selective NMDA receptor non-competitive antagonist (IC50 values are 3, 6, 229, and >300, >300 μM for NR2D, NR2C, NR2A, NR2B, and GluR1, respectively).
Product name: QNZ46 | Cat No. DC8307 |Cas: 1237744-13-6 |Other names: QNZ-46,QNZ 46,QNZ46 |Molecule formular: C24H17N3O6 |Molecule Weight: 443.41 |Purity>98%
QNZ is a NR2C/NR2D-selective NMDA receptor non-competitive antagonist (IC50 values are 3, 6, 229, and >300, >300 μM for NR2D, NR2C, NR2A, NR2B, and GluR1, respectively).
For research and scientific purpose only, not for human use.
QNZ is a NR2C/NR2D-selective NMDA receptor non-competitive antagonist (IC50 values are 3, 6, 229, and >300, >300 μM for NR2D, NR2C, NR2A, NR2B, and GluR1, respectively).
Product name: QNZ46 | Cat No. DC8307 |Cas: 1237744-13-6 |Other names: QNZ-46,QNZ 46,QNZ46 |Molecule formular: C24H17N3O6 |Molecule Weight: 443.41 |Purity>98%
QNZ is a NR2C/NR2D-selective NMDA receptor non-competitive antagonist (IC50 values are 3, 6, 229, and >300, >300 μM for NR2D, NR2C, NR2A, NR2B, and GluR1, respectively).
For research and scientific purpose only, not for human use.
RQ-00203078| TRPM8 inhibitor|DC Chemicals
RQ-00203078| TRPM8 inhibitor|DC Chemicals
RQ-00203078 is a potent TRPM8 antagonist (IC50 values are 5.3 and 8.3 nM for rat and human channels respectively).
Product name: RQ-00203078 | Cat No. DC8306 |Cas: 1254205-52-1 |Other names: |Molecule formular: C21H13ClF6N2O5S |Molecule Weight: 554.85 |Purity>98%
RQ-00203078 is a potent TRPM8 antagonist (IC50 values are 5.3 and 8.3 nM for rat and human channels respectively).
For research and scientific purpose only, not for human use.
RQ-00203078 is a potent TRPM8 antagonist (IC50 values are 5.3 and 8.3 nM for rat and human channels respectively).
Product name: RQ-00203078 | Cat No. DC8306 |Cas: 1254205-52-1 |Other names: |Molecule formular: C21H13ClF6N2O5S |Molecule Weight: 554.85 |Purity>98%
RQ-00203078 is a potent TRPM8 antagonist (IC50 values are 5.3 and 8.3 nM for rat and human channels respectively).
For research and scientific purpose only, not for human use.
Edoxaban|CAS 912273-65-5|DC Chemicals
Edoxaban|CAS 912273-65-5|DC Chemicals
Edoxaban(DU-176) is an oral factor Xa (FXa) inhibitor in clinical development for stroke prevention
Product name: Edoxaban | Cat No. DC8305 |Cas: 912273-65-5 |Other names: |Molecule formular: C24H30ClN7O4S |Molecule Weight: 548.1 |Purity>98%
Edoxaban(DU-176) is an oral factor Xa (FXa) inhibitor in clinical development for stroke prevention
For research and scientific purpose only, not for human use.
Edoxaban(DU-176) is an oral factor Xa (FXa) inhibitor in clinical development for stroke prevention
Product name: Edoxaban | Cat No. DC8305 |Cas: 912273-65-5 |Other names: |Molecule formular: C24H30ClN7O4S |Molecule Weight: 548.1 |Purity>98%
Edoxaban(DU-176) is an oral factor Xa (FXa) inhibitor in clinical development for stroke prevention
For research and scientific purpose only, not for human use.
Isoxazole 9(ISX9)|Neuronal Differentiation Inducer|DC Chemicals
Isoxazole 9(ISX9)|Neuronal Differentiation Inducer|DC Chemicals
ISX-9 is a small molecule inducer of adult neural stem cell differentiation both in vitro and in vivo.
Product name: Isoxazole 9(ISX9) | Cat No. DC8304 |Cas: 832115-62-5 |Other names: ISX-9,ISX 9,Neuronal Differentiation Inducer III |Molecule formular: C11H10N2O2S |Molecule Weight: 234.3 |Purity>98%
ISX-9 is a small molecule inducer of adult neural stem cell differentiation both in vitro and in vivo.
For research and scientific purpose only, not for human use.
ISX-9 is a small molecule inducer of adult neural stem cell differentiation both in vitro and in vivo.
Product name: Isoxazole 9(ISX9) | Cat No. DC8304 |Cas: 832115-62-5 |Other names: ISX-9,ISX 9,Neuronal Differentiation Inducer III |Molecule formular: C11H10N2O2S |Molecule Weight: 234.3 |Purity>98%
ISX-9 is a small molecule inducer of adult neural stem cell differentiation both in vitro and in vivo.
For research and scientific purpose only, not for human use.
GTS 21 2HCl(DMXBA)|CAS 156223-05-1|DC Chemicals
GTS 21 2HCl(DMXBA)|CAS 156223-05-1|DC Chemicals
GTS 21 dihydrochloride is a partial agonist of α7 nicotinic acetylcholine receptors (nAChRs); also a weak α4β2 and 5-HT3 antagonist at micromolar concentrations.
Product name: GTS 21 2HCl(DMXBA) | Cat No. DC8303 |Cas: 156223-05-1 |Other names: GTS21,GTS 21,GTS-21 |Molecule formular: C19H20N2O2.2HCl |Molecule Weight: 381.3 |Purity>98%
GTS 21 dihydrochloride is a partial agonist of α7 nicotinic acetylcholine receptors (nAChRs); also a weak α4β2 and 5-HT3 antagonist at micromolar concentrations.
For research and scientific purpose only, not for human use.
GTS 21 dihydrochloride is a partial agonist of α7 nicotinic acetylcholine receptors (nAChRs); also a weak α4β2 and 5-HT3 antagonist at micromolar concentrations.
Product name: GTS 21 2HCl(DMXBA) | Cat No. DC8303 |Cas: 156223-05-1 |Other names: GTS21,GTS 21,GTS-21 |Molecule formular: C19H20N2O2.2HCl |Molecule Weight: 381.3 |Purity>98%
GTS 21 dihydrochloride is a partial agonist of α7 nicotinic acetylcholine receptors (nAChRs); also a weak α4β2 and 5-HT3 antagonist at micromolar concentrations.
For research and scientific purpose only, not for human use.
Elacridar |P-glycoprotein (P-gp/ABCG1) inhibitor|DC Chemicals
Elacridar |P-glycoprotein (P-gp/ABCG1) inhibitor|DC Chemicals
Elacridar hydrochloride is an orally selectly potent P-glycoprotein (P-gp/ABCG1) inhibitor.
Product name: Elacridar hydrochloride | Cat No. DC8301 |Cas: 143851-98-3，143664-11-3（free base） |Other names: GF 120918,GF120918,GF-120918 |Molecule formular: C34H33N3O5.HCl |Molecule Weight: 600.1 |Purity>98%
Elacridar hydrochloride is an orally selectly potent P-glycoprotein (P-gp/ABCG1) inhibitor.
For research and scientific purpose only, not for human use.
Elacridar hydrochloride is an orally selectly potent P-glycoprotein (P-gp/ABCG1) inhibitor.
Product name: Elacridar hydrochloride | Cat No. DC8301 |Cas: 143851-98-3，143664-11-3（free base） |Other names: GF 120918,GF120918,GF-120918 |Molecule formular: C34H33N3O5.HCl |Molecule Weight: 600.1 |Purity>98%
Elacridar hydrochloride is an orally selectly potent P-glycoprotein (P-gp/ABCG1) inhibitor.
For research and scientific purpose only, not for human use.
Entrectinib (RXDX-101)|ALK inhibit|DC Chemicals
Entrectinib (RXDX-101)|ALK inhibit|DC Chemicals
Entrectinib (RXDX-101), a potent and selective small molecule inhibitor of TrkA/B/C, ROS1, and ALK kinases, has demonstrated early clinical activity when orally administered intermittently under fasting conditions.
Product name: Entrectinib (RXDX-101) | Cat No. DC8300 |Cas: 1108743-60-7 |Other names: NMS E628; RXDX-101,NMSE628; RXDX 101,NMS-E628; RXDX101 |Molecule formular: C31H34F2N6O2 |Molecule Weight: 560.64 |Purity>98%
Entrectinib (RXDX-101), a potent and selective small molecule inhibitor of TrkA/B/C, ROS1, and ALK kinases, has demonstrated early clinical activity when orally administered intermittently under fasting conditions.
For research and scientific purpose only, not for human use.
Entrectinib (RXDX-101), a potent and selective small molecule inhibitor of TrkA/B/C, ROS1, and ALK kinases, has demonstrated early clinical activity when orally administered intermittently under fasting conditions.
Product name: Entrectinib (RXDX-101) | Cat No. DC8300 |Cas: 1108743-60-7 |Other names: NMS E628; RXDX-101,NMSE628; RXDX 101,NMS-E628; RXDX101 |Molecule formular: C31H34F2N6O2 |Molecule Weight: 560.64 |Purity>98%
Entrectinib (RXDX-101), a potent and selective small molecule inhibitor of TrkA/B/C, ROS1, and ALK kinases, has demonstrated early clinical activity when orally administered intermittently under fasting conditions.
For research and scientific purpose only, not for human use.
BAN ORL 24|BAN ORL24|ORL1 agonist|DC Chemicals
BAN ORL 24|BAN ORL24|ORL1 agonist|DC Chemicals
BAN ORL 24 is a potent, selective, competitive ORL1 non-peptide agonist. Displays 1000-fold selectivity over classical opioid receptors.
Product name: BAN ORL 24 | Cat No. DC8298 |Cas: 1401463-54-4 |Other names: BANORL 24,BAN ORL24,BANORL24,BAN ORL-24 |Molecule formular: C27H35N3O2.2HCl |Molecule Weight: 506.51 |Purity>98%
BAN ORL 24 is a potent, selective, competitive ORL1 non-peptide agonist. Displays 1000-fold selectivity over classical opioid receptors.
For research and scientific purpose only, not for human use.
BAN ORL 24 is a potent, selective, competitive ORL1 non-peptide agonist. Displays 1000-fold selectivity over classical opioid receptors.
Product name: BAN ORL 24 | Cat No. DC8298 |Cas: 1401463-54-4 |Other names: BANORL 24,BAN ORL24,BANORL24,BAN ORL-24 |Molecule formular: C27H35N3O2.2HCl |Molecule Weight: 506.51 |Purity>98%
BAN ORL 24 is a potent, selective, competitive ORL1 non-peptide agonist. Displays 1000-fold selectivity over classical opioid receptors.
For research and scientific purpose only, not for human use.
ZM 39923|ZM39923|JAK3 inhibitor|DC Chemicals
ZM 39923|ZM39923|JAK3 inhibitor|DC Chemicals
ZM 39923 is an inhibitor of JAK3 (IC50 = 79 nM) that less potently inhibits epidermal growth factor receptor, JAK1, and cyclin-dependent kinase 4 (IC50s = 2.4, 40, and 10 µM, respectively).
Product name: ZM 39923 hydrochloride | Cat No. DC8297 |Cas: 1021868-92-7 |Other names: ZM 39923,ZM39923,ZM-39923 |Molecule formular: C23H26ClNO |Molecule Weight: 367.91 |Purity>98%
ZM 39923 is an inhibitor of JAK3 (IC50 = 79 nM) that less potently inhibits epidermal growth factor receptor, JAK1, and cyclin-dependent kinase 4 (IC50s = 2.4, 40, and 10 µM, respectively).
For research and scientific purpose only, not for human use.
ZM 39923 is an inhibitor of JAK3 (IC50 = 79 nM) that less potently inhibits epidermal growth factor receptor, JAK1, and cyclin-dependent kinase 4 (IC50s = 2.4, 40, and 10 µM, respectively).
Product name: ZM 39923 hydrochloride | Cat No. DC8297 |Cas: 1021868-92-7 |Other names: ZM 39923,ZM39923,ZM-39923 |Molecule formular: C23H26ClNO |Molecule Weight: 367.91 |Purity>98%
ZM 39923 is an inhibitor of JAK3 (IC50 = 79 nM) that less potently inhibits epidermal growth factor receptor, JAK1, and cyclin-dependent kinase 4 (IC50s = 2.4, 40, and 10 µM, respectively).
For research and scientific purpose only, not for human use.
Dorsomorphin|BML275|AMPK INHIBITOR|DC Chemicals
Dorsomorphin|BML275|AMPK INHIBITOR|DC Chemicals
Dorsomorphin(Compound C; BML-275) has been shown to act as a potent and selective inhibitor of AMPK (AMP-activated protein kinase; Ki = 109 nM), induced by AICAR and metformin; also inhibits the bone morphogenetic protein type 1 receptors ACTR-I (ALK2), BMPR-IA (ALK3), and BMPR-IB (ALK 6).
Product name: Dorsomorphin(BML-275) | Cat No. DC8296 |Cas: 866405-64-3 |Other names: BML-275; Compound C; BML275; BML 275 |Molecule formular: C24H25N5O |Molecule Weight: 399.49 |Purity>98%
Dorsomorphin(Compound C; BML-275) has been shown to act as a potent and selective inhibitor of AMPK (AMP-activated protein kinase; Ki = 109 nM), induced by AICAR and metformin; also inhibits the bone morphogenetic protein type 1 receptors ACTR-I (ALK2), BMPR-IA (ALK3), and BMPR-IB (ALK 6).
For research and scientific purpose only, not for human use.
Dorsomorphin(Compound C; BML-275) has been shown to act as a potent and selective inhibitor of AMPK (AMP-activated protein kinase; Ki = 109 nM), induced by AICAR and metformin; also inhibits the bone morphogenetic protein type 1 receptors ACTR-I (ALK2), BMPR-IA (ALK3), and BMPR-IB (ALK 6).
Product name: Dorsomorphin(BML-275) | Cat No. DC8296 |Cas: 866405-64-3 |Other names: BML-275; Compound C; BML275; BML 275 |Molecule formular: C24H25N5O |Molecule Weight: 399.49 |Purity>98%
Dorsomorphin(Compound C; BML-275) has been shown to act as a potent and selective inhibitor of AMPK (AMP-activated protein kinase; Ki = 109 nM), induced by AICAR and metformin; also inhibits the bone morphogenetic protein type 1 receptors ACTR-I (ALK2), BMPR-IA (ALK3), and BMPR-IB (ALK 6).
For research and scientific purpose only, not for human use.
trans-Tranilast|cas 70806-55-2|DC Chemicals
trans-Tranilast|cas 70806-55-2|DC Chemicals
trans-Tranilast
Product name: trans-Tranilast | Cat No. DC8295 |Cas: 70806-55-2 |Other names: |Molecule formular: C18H17NO5 |Molecule Weight: 327.33 |Purity>98%
For research and scientific purpose only, not for human use.
trans-Tranilast
Product name: trans-Tranilast | Cat No. DC8295 |Cas: 70806-55-2 |Other names: |Molecule formular: C18H17NO5 |Molecule Weight: 327.33 |Purity>98%
For research and scientific purpose only, not for human use.
BPR1J-097|FLT-3 Inhibitor|DC Chemicals
BPR1J-097|FLT-3 Inhibitor|DC Chemicals
BPR1J-097 is a novel small molecule FLT-3 inhibitor(IC50=11±7 nM) with promising in vivo anti-tumour activities; inhibits FLT-3 D835Y with an IC50 of 3 nM.
Product name: BPR1J-097 | Cat No. DC8294 |Cas: 1327167-19-0 |Other names: BPR1J-097，BPR1J 097，BPR1J097 |Molecule formular: C27H28N6O3S |Molecule Weight: 516.61 |Purity>98%
BPR1J-097 is a novel small molecule FLT-3 inhibitor(IC50=11±7 nM) with promising in vivo anti-tumour activities; inhibits FLT-3 D835Y with an IC50 of 3 nM.
For research and scientific purpose only, not for human use.
BPR1J-097 is a novel small molecule FLT-3 inhibitor(IC50=11±7 nM) with promising in vivo anti-tumour activities; inhibits FLT-3 D835Y with an IC50 of 3 nM.
Product name: BPR1J-097 | Cat No. DC8294 |Cas: 1327167-19-0 |Other names: BPR1J-097，BPR1J 097，BPR1J097 |Molecule formular: C27H28N6O3S |Molecule Weight: 516.61 |Purity>98%
BPR1J-097 is a novel small molecule FLT-3 inhibitor(IC50=11±7 nM) with promising in vivo anti-tumour activities; inhibits FLT-3 D835Y with an IC50 of 3 nM.
For research and scientific purpose only, not for human use.
2015年9月16日星期三
UNC-0224|UNC0224|PRMTs inhibitor|DC Chemicals
UNC-0224|UNC0224|PRMTs inhibitor|DC Chemicals
UNC-0224 is a potent inhibitor of G9a histone lysine methyltransferase (IC50 = 15 nM).
Product name: UNC-0224 | Cat No. DC8293 |Cas: 1197196-48-7 |Other names: UNC-0224, UNC0224, UNC 0224 |Molecule formular: C26H43N7O2 |Molecule Weight: 485.67 |Purity>98%
UNC-0224 is a potent inhibitor of G9a histone lysine methyltransferase (IC50 = 15 nM).
For research and scientific purpose only, not for human use.
UNC-0224 is a potent inhibitor of G9a histone lysine methyltransferase (IC50 = 15 nM).
Product name: UNC-0224 | Cat No. DC8293 |Cas: 1197196-48-7 |Other names: UNC-0224, UNC0224, UNC 0224 |Molecule formular: C26H43N7O2 |Molecule Weight: 485.67 |Purity>98%
UNC-0224 is a potent inhibitor of G9a histone lysine methyltransferase (IC50 = 15 nM).
For research and scientific purpose only, not for human use.
AMI-1|PRMT inhibitor| DC Chemicals
AMI-1|PRMT inhibitor| DC Chemicals
AMI-1 is a PRMT and HIV-1 RT polymerase inhibitor.
Product name: AMI-1 | Cat No. DC8292 |Cas: 20324-87-2 |Other names: AMI-1,AMI 1,AMI1 |Molecule formular: C21H12N2O9S2•4Na |Molecule Weight: 592.42 |Purity>98%
AMI-1 is a PRMT and HIV-1 RT polymerase inhibitor.
For research and scientific purpose only, not for human use.
AMI-1 is a PRMT and HIV-1 RT polymerase inhibitor.
Product name: AMI-1 | Cat No. DC8292 |Cas: 20324-87-2 |Other names: AMI-1,AMI 1,AMI1 |Molecule formular: C21H12N2O9S2•4Na |Molecule Weight: 592.42 |Purity>98%
AMI-1 is a PRMT and HIV-1 RT polymerase inhibitor.
For research and scientific purpose only, not for human use.
PFI-4|BRPF1 bromodomain inhibitor| DC Chemicals
PFI-4|BRPF1 bromodomain inhibitor| DC Chemicals
PFI-4 is a potent and selective BRPF1 bromodomain inhibitor (IC50 = 80 nM).
Product name: PFI-4 | Cat No. DC8291 |Cas: 900305-37-5 |Other names: PFI4，PFI 4 |Molecule formular: C21H24N4O3 |Molecule Weight: 380.44 |Purity>98%
PFI-4 is a potent and selective BRPF1 bromodomain inhibitor (IC50 = 80 nM).
For research and scientific purpose only, not for human use.
PFI-4 is a potent and selective BRPF1 bromodomain inhibitor (IC50 = 80 nM).
Product name: PFI-4 | Cat No. DC8291 |Cas: 900305-37-5 |Other names: PFI4，PFI 4 |Molecule formular: C21H24N4O3 |Molecule Weight: 380.44 |Purity>98%
PFI-4 is a potent and selective BRPF1 bromodomain inhibitor (IC50 = 80 nM).
For research and scientific purpose only, not for human use.
S-PFI-2 HCl|Negative of R-PFI-2| DC Chemicals
S-PFI-2 HCl|Negative of R-PFI-2| DC Chemicals
Negative control of (R)-PFI 2 hydrochloride. Exhibits 500-fold lower activity in a SETD7 enzymatic assay (IC50 = 1 μM) compared to the active enantiomer.
Product name: S-PFI-2(HCl) | Cat No. DC8290 |Cas: N/A |Other names: PFI2,PFI-2,SPFI2,SPFI-2,PFI 2,SPFI 2 |Molecule formular: C23H25F4N3O3S.HCl |Molecule Weight: 535.98 |Purity>98%
Negative control of (R)-PFI 2 hydrochloride. Exhibits 500-fold lower activity in a SETD7 enzymatic assay (IC50 = 1 μM) compared to the active enantiomer.
For research and scientific purpose only, not for human use.
Negative control of (R)-PFI 2 hydrochloride. Exhibits 500-fold lower activity in a SETD7 enzymatic assay (IC50 = 1 μM) compared to the active enantiomer.
Product name: S-PFI-2(HCl) | Cat No. DC8290 |Cas: N/A |Other names: PFI2,PFI-2,SPFI2,SPFI-2,PFI 2,SPFI 2 |Molecule formular: C23H25F4N3O3S.HCl |Molecule Weight: 535.98 |Purity>98%
Negative control of (R)-PFI 2 hydrochloride. Exhibits 500-fold lower activity in a SETD7 enzymatic assay (IC50 = 1 μM) compared to the active enantiomer.
For research and scientific purpose only, not for human use.
VER155008|VER-155008|cas 1134156-31-2| DC Chemicals
VER155008|VER-155008|cas 1134156-31-2| DC Chemicals
VER-155008 is a novel, small molecule inhibitor of Hsc70/Hsp70 with GI50 of 5.3-14.4 uM in human breast and colon cancer cell lines.
Product name: VER155008 | Cat No. DC8299 |Cas: 1134156-31-2 |Other names: VER 155008,VER-155008,VER155008 |Molecule formular: C25H23Cl2N7O4 |Molecule Weight: 556.4 |Purity>98%
VER-155008 is a novel, small molecule inhibitor of Hsc70/Hsp70 with GI50 of 5.3-14.4 uM in human breast and colon cancer cell lines.
For research and scientific purpose only, not for human use.
VER-155008 is a novel, small molecule inhibitor of Hsc70/Hsp70 with GI50 of 5.3-14.4 uM in human breast and colon cancer cell lines.
Product name: VER155008 | Cat No. DC8299 |Cas: 1134156-31-2 |Other names: VER 155008,VER-155008,VER155008 |Molecule formular: C25H23Cl2N7O4 |Molecule Weight: 556.4 |Purity>98%
VER-155008 is a novel, small molecule inhibitor of Hsc70/Hsp70 with GI50 of 5.3-14.4 uM in human breast and colon cancer cell lines.
For research and scientific purpose only, not for human use.
Ramatroban (BAY u3405)|cas 116649-85-5| DC Chemicals
Ramatroban (BAY u3405)|cas 116649-85-5| DC Chemicals
Ramatroban (BAY u3405) is a thromboxane A(2) (TxA(2)) antagonist marketed for allergic rhinitis.
Product name: Ramatroban (BAY u3405) | Cat No. DC6918 |Cas: 116649-85-5 |Other names: BAY u3405; BAY-u3405 |Molecule formular: C21H21FN2O4S |Molecule Weight: 416.47 |Purity>98%
Ramatroban (BAY u3405) is a thromboxane A(2) (TxA(2)) antagonist marketed for allergic rhinitis.
For research and scientific purpose only, not for human use.
Ramatroban (BAY u3405) is a thromboxane A(2) (TxA(2)) antagonist marketed for allergic rhinitis.
Product name: Ramatroban (BAY u3405) | Cat No. DC6918 |Cas: 116649-85-5 |Other names: BAY u3405; BAY-u3405 |Molecule formular: C21H21FN2O4S |Molecule Weight: 416.47 |Purity>98%
Ramatroban (BAY u3405) is a thromboxane A(2) (TxA(2)) antagonist marketed for allergic rhinitis.
For research and scientific purpose only, not for human use.
Vonoprazan|cas 881681-00-1|DC Chemicals
Vonoprazan|cas 881681-00-1|DC Chemicals
Product name: Vonoprazan | Cat No. DC6917 |Cas: 881681-00-1 |Other names: 1-[5-(2-Fluorophenyl)-1-[(pyridin-3-yl)sulfonyl]-1H-pyrrol-3-yl]-N-methylmethanamine
|Molecule formular: C17H16FN3O2S |Molecule Weight: 345.3912432 |Purity>98%
For research and scientific purpose only, not for human use.
Product name: Vonoprazan | Cat No. DC6917 |Cas: 881681-00-1 |Other names: 1-[5-(2-Fluorophenyl)-1-[(pyridin-3-yl)sulfonyl]-1H-pyrrol-3-yl]-N-methylmethanamine
|Molecule formular: C17H16FN3O2S |Molecule Weight: 345.3912432 |Purity>98%
For research and scientific purpose only, not for human use.
Zucapsaicin|cas 25775-90-0|DC Chemicals
Zucapsaicin|cas 25775-90-0|DC Chemicals
Product name: Zucapsaicin | Cat No. DC6916 |Cas: 25775-90-0 |Other names: Zucapsaicin,cis-capsaicin,civamide,(Z)-CAPSAICIN |Molecule formular: C18H27NO3 |Molecule Weight: 305.41 |Purity>98%
For research and scientific purpose only, not for human use.
Product name: Zucapsaicin | Cat No. DC6916 |Cas: 25775-90-0 |Other names: Zucapsaicin,cis-capsaicin,civamide,(Z)-CAPSAICIN |Molecule formular: C18H27NO3 |Molecule Weight: 305.41 |Purity>98%
For research and scientific purpose only, not for human use.
Phenothrin|cas 26002-80-2|DC Chemicals
Phenothrin|cas 26002-80-2|DC Chemicals
Product name: Phenothrin | Cat No. DC6915 |Cas: 26002-80-2 |Other names: (+)-(z,e)-leste |Molecule formular: C23H26O3 |Molecule Weight: 350.45 |Purity>98%
For research and scientific purpose only, not for human use.
Product name: Phenothrin | Cat No. DC6915 |Cas: 26002-80-2 |Other names: (+)-(z,e)-leste |Molecule formular: C23H26O3 |Molecule Weight: 350.45 |Purity>98%
For research and scientific purpose only, not for human use.
Trelagliptin(SYR-472)|DC Chemicals
Trelagliptin(SYR-472)|DC Chemicals
Trelagliptin(SYR-472) is a long acting dipeptidyl peptidase-4 (DPP-4) inhibitor that is being developed for the treatment of type 2 diabetes (T2D).
Product name: Trelagliptin(SYR-472) | Cat No. DC6914 |Cas: 1029877-94-8 |Other names: SYR-472 succinate; SYR472 succinate; SYR 472 succinate |Molecule formular: C22H26FN5O6 |Molecule Weight: 475.47 |Purity>98%
Trelagliptin(SYR-472) is a long acting dipeptidyl peptidase-4 (DPP-4) inhibitor that is being developed for the treatment of type 2 diabetes (T2D).
For research and scientific purpose only, not for human use.
Trelagliptin(SYR-472) is a long acting dipeptidyl peptidase-4 (DPP-4) inhibitor that is being developed for the treatment of type 2 diabetes (T2D).
Product name: Trelagliptin(SYR-472) | Cat No. DC6914 |Cas: 1029877-94-8 |Other names: SYR-472 succinate; SYR472 succinate; SYR 472 succinate |Molecule formular: C22H26FN5O6 |Molecule Weight: 475.47 |Purity>98%
Trelagliptin(SYR-472) is a long acting dipeptidyl peptidase-4 (DPP-4) inhibitor that is being developed for the treatment of type 2 diabetes (T2D).
For research and scientific purpose only, not for human use.
Efaproxiral|cas 131179-95-8| DC Chemicals
Efaproxiral|cas 131179-95-8| DC Chemicals
Product name: Efaproxiral | Cat No. DC6913 |Cas: 131179-95-8 |Other names: Efaproxiral，Efaproxiral free acid，faproxiral |Molecule formular: C20H22NO4.Na |Molecule Weight: 341.4 |Purity>98%
For research and scientific purpose only, not for human use.
Product name: Efaproxiral | Cat No. DC6913 |Cas: 131179-95-8 |Other names: Efaproxiral，Efaproxiral free acid，faproxiral |Molecule formular: C20H22NO4.Na |Molecule Weight: 341.4 |Purity>98%
For research and scientific purpose only, not for human use.
Ethofibrate|DC Chemicals
Ethofibrate|DC Chemicals
Product name: Ethofibrate | Cat No. DC6912 |Cas: 31637-97-5 |Other names: Ethofibrate，Lipo-merz，XE-14-543，Tricerol |Molecule formular: C18H18ClNO5 |Molecule Weight: 363.79 |Purity>98%
For research and scientific purpose only, not for human use.
Product name: Ethofibrate | Cat No. DC6912 |Cas: 31637-97-5 |Other names: Ethofibrate，Lipo-merz，XE-14-543，Tricerol |Molecule formular: C18H18ClNO5 |Molecule Weight: 363.79 |Purity>98%
For research and scientific purpose only, not for human use.
pardoprunox (SLV308)|DC Chemicals
pardoprunox (SLV308)|DC Chemicals
Pardoprunox(SLV-308) is a novel partial dopamine D2 and D3 receptor agonist and serotonin 5-HT1A receptor agonist; D2 (pKi = 8.1) and D3 receptor (pKi = 8.6) partial agonist (IA = 50% and 67%, respectively) and 5-HT1A receptor (pKi = 8.5) full agonist (IA = 100%). It also binds to D4 (pKi = 7.8), α1-adrenergic (pKi = 7.8), α2-adrenergic (pKi = 7.4), and 5-HT7 receptors (pKi = 7.2) with lower affinity.
Product name: pardoprunox (SLV308) | Cat No. DC6911 |Cas: 269718-84-5 |Other names: SLV-308; DU-126891 |Molecule formular: C12H15N3O2 |Molecule Weight: 233.27 |Purity>98%
Pardoprunox(SLV-308) is a novel partial dopamine D2 and D3 receptor agonist and serotonin 5-HT1A receptor agonist; D2 (pKi = 8.1) and D3 receptor (pKi = 8.6) partial agonist (IA = 50% and 67%, respectively) and 5-HT1A receptor (pKi = 8.5) full agonist (IA = 100%). It also binds to D4 (pKi = 7.8), α1-adrenergic (pKi = 7.8), α2-adrenergic (pKi = 7.4), and 5-HT7 receptors (pKi = 7.2) with lower affinity.
For research and scientific purpose only, not for human use.
Pardoprunox(SLV-308) is a novel partial dopamine D2 and D3 receptor agonist and serotonin 5-HT1A receptor agonist; D2 (pKi = 8.1) and D3 receptor (pKi = 8.6) partial agonist (IA = 50% and 67%, respectively) and 5-HT1A receptor (pKi = 8.5) full agonist (IA = 100%). It also binds to D4 (pKi = 7.8), α1-adrenergic (pKi = 7.8), α2-adrenergic (pKi = 7.4), and 5-HT7 receptors (pKi = 7.2) with lower affinity.
Product name: pardoprunox (SLV308) | Cat No. DC6911 |Cas: 269718-84-5 |Other names: SLV-308; DU-126891 |Molecule formular: C12H15N3O2 |Molecule Weight: 233.27 |Purity>98%
Pardoprunox(SLV-308) is a novel partial dopamine D2 and D3 receptor agonist and serotonin 5-HT1A receptor agonist; D2 (pKi = 8.1) and D3 receptor (pKi = 8.6) partial agonist (IA = 50% and 67%, respectively) and 5-HT1A receptor (pKi = 8.5) full agonist (IA = 100%). It also binds to D4 (pKi = 7.8), α1-adrenergic (pKi = 7.8), α2-adrenergic (pKi = 7.4), and 5-HT7 receptors (pKi = 7.2) with lower affinity.
For research and scientific purpose only, not for human use.
NS-1643|NS1643|DC Chemicals
NS-1643|NS1643|DC Chemicals
NS1643 is a potent human ether-a-go-go related gene (hERG) KV11.1 channel activator (EC50 = 10.5 μM).
Product name: NS-1643 | Cat No. DC6910 |Cas: 448895-37-2 |Other names: NS-1643 |Molecule formular: C15H10F6N2O3 |Molecule Weight: 380.24 |Purity>98%
NS1643 is a potent human ether-a-go-go related gene (hERG) KV11.1 channel activator (EC50 = 10.5 μM).
For research and scientific purpose only, not for human use.
NS1643 is a potent human ether-a-go-go related gene (hERG) KV11.1 channel activator (EC50 = 10.5 μM).
Product name: NS-1643 | Cat No. DC6910 |Cas: 448895-37-2 |Other names: NS-1643 |Molecule formular: C15H10F6N2O3 |Molecule Weight: 380.24 |Purity>98%
NS1643 is a potent human ether-a-go-go related gene (hERG) KV11.1 channel activator (EC50 = 10.5 μM).
For research and scientific purpose only, not for human use.
Prucalopride succinate|DC Chemicals
Prucalopride succinate|DC Chemicals
Prucalopride succinate is a selective, high affinity 5-HT4 receptor agonist with pKi of 8.6/8.1 for 5-HT4a/4b.
Product name: Prucalopride succinate | Cat No. DC8289 |Cas: 179474-85-2 |Other names: Resolor; R-108512 |Molecule formular: C22H32ClN3O7 |Molecule Weight: 485.96 |Purity>98%
Prucalopride succinate is a selective, high affinity 5-HT4 receptor agonist with pKi of 8.6/8.1 for 5-HT4a/4b.
For research and scientific purpose only, not for human use.
Prucalopride succinate is a selective, high affinity 5-HT4 receptor agonist with pKi of 8.6/8.1 for 5-HT4a/4b.
Product name: Prucalopride succinate | Cat No. DC8289 |Cas: 179474-85-2 |Other names: Resolor; R-108512 |Molecule formular: C22H32ClN3O7 |Molecule Weight: 485.96 |Purity>98%
Prucalopride succinate is a selective, high affinity 5-HT4 receptor agonist with pKi of 8.6/8.1 for 5-HT4a/4b.
For research and scientific purpose only, not for human use.
Vortioxetine(Lu AA21004)|DC Chemicals
Vortioxetine(Lu AA21004)|DC Chemicals
Vortioxetine Hcl (Lu AA21004 Hcl) is a multimodal serotonergic agent, inhibits 5-HT1A, 5-HT1B, 5-HT3A, 5-HT7 receptor and SERT with IC50 of 15 nM, 33 nM, 3.7 nM, 19 nM and 1.6 nM, respectively.
Product name: Vortioxetine hydrobromide | Cat No. DC8288 |Cas: 960203-27-4 |Other names: Lu AA 21004 hydrobromide; Lu AA21004 hydrobromide |Molecule formular: C18H23BrN2S |Molecule Weight: 379.36 |Purity>98%
Vortioxetine Hcl (Lu AA21004 Hcl) is a multimodal serotonergic agent, inhibits 5-HT1A, 5-HT1B, 5-HT3A, 5-HT7 receptor and SERT with IC50 of 15 nM, 33 nM, 3.7 nM, 19 nM and 1.6 nM, respectively.
For research and scientific purpose only, not for human use.
Vortioxetine Hcl (Lu AA21004 Hcl) is a multimodal serotonergic agent, inhibits 5-HT1A, 5-HT1B, 5-HT3A, 5-HT7 receptor and SERT with IC50 of 15 nM, 33 nM, 3.7 nM, 19 nM and 1.6 nM, respectively.
Product name: Vortioxetine hydrobromide | Cat No. DC8288 |Cas: 960203-27-4 |Other names: Lu AA 21004 hydrobromide; Lu AA21004 hydrobromide |Molecule formular: C18H23BrN2S |Molecule Weight: 379.36 |Purity>98%
Vortioxetine Hcl (Lu AA21004 Hcl) is a multimodal serotonergic agent, inhibits 5-HT1A, 5-HT1B, 5-HT3A, 5-HT7 receptor and SERT with IC50 of 15 nM, 33 nM, 3.7 nM, 19 nM and 1.6 nM, respectively.
For research and scientific purpose only, not for human use.
Lubiprostone|DC Chemicals
Lubiprostone|DC Chemicals
Product name: Lubiprostone | Cat No. DC8287 |Cas: 333963-40-9 |Other names: Spi 0211，Unii-7662kg2R6k，AMitiza Lubiprostone |Molecule formular: C20H32F2O5 |Molecule Weight: 390.46 |Purity>98%
For research and scientific purpose only, not for human use.
Product name: Lubiprostone | Cat No. DC8287 |Cas: 333963-40-9 |Other names: Spi 0211，Unii-7662kg2R6k，AMitiza Lubiprostone |Molecule formular: C20H32F2O5 |Molecule Weight: 390.46 |Purity>98%
For research and scientific purpose only, not for human use.
Brexpiprazole(OPC34712)|D2 dopamine partial agonist|DC Chemicals
Brexpiprazole(OPC34712)|D2 dopamine partial agonist|DC Chemicals
Brexpiprazole is a novel D2 dopamine partial agonist.
Product name: Brexpiprazole(OPC34712) | Cat No. DC8286 |Cas: 913611-97-9 |Other names: OPC 34712; OPC34712; OPC-34712 |Molecule formular: C25H27N3O2S |Molecule Weight: 433.57 |Purity>98%
Brexpiprazole is a novel D2 dopamine partial agonist.
For research and scientific purpose only, not for human use.
Brexpiprazole is a novel D2 dopamine partial agonist.
Product name: Brexpiprazole(OPC34712) | Cat No. DC8286 |Cas: 913611-97-9 |Other names: OPC 34712; OPC34712; OPC-34712 |Molecule formular: C25H27N3O2S |Molecule Weight: 433.57 |Purity>98%
Brexpiprazole is a novel D2 dopamine partial agonist.
For research and scientific purpose only, not for human use.
Acotiamide HCl|DC Chemicals
Acotiamide HCl|DC Chemicals
Product name: Acotiamide HCl | Cat No. DC8285 |Cas: 773092-05-0 |Other names: Ym-443，Acotiamide HCl |Molecule formular: C21H31ClN4O5S |Molecule Weight: 487.013 |Purity>98%
For research and scientific purpose only, not for human use.
Product name: Acotiamide HCl | Cat No. DC8285 |Cas: 773092-05-0 |Other names: Ym-443，Acotiamide HCl |Molecule formular: C21H31ClN4O5S |Molecule Weight: 487.013 |Purity>98%
For research and scientific purpose only, not for human use.
Almotriptan Malate(PNU180638)|cas 181183-52-8|DC Chemicals
Almotriptan Malate(PNU180638)|cas 181183-52-8|DC Chemicals
Almotriptan Malate is a 5-HT1B/1D-receptor agonist used to treat migraine.
Product name: Almotriptan Malate(PNU180638) | Cat No. DC8284 |Cas: 181183-52-8 |Other names: Axert; Almogran; PNU-180638,PNU 180638 |Molecule formular: C21H31N3O7S |Molecule Weight: 469.55 |Purity>98%
Almotriptan Malate is a 5-HT1B/1D-receptor agonist used to treat migraine.
For research and scientific purpose only, not for human use.
Almotriptan Malate is a 5-HT1B/1D-receptor agonist used to treat migraine.
Product name: Almotriptan Malate(PNU180638) | Cat No. DC8284 |Cas: 181183-52-8 |Other names: Axert; Almogran; PNU-180638,PNU 180638 |Molecule formular: C21H31N3O7S |Molecule Weight: 469.55 |Purity>98%
Almotriptan Malate is a 5-HT1B/1D-receptor agonist used to treat migraine.
For research and scientific purpose only, not for human use.
PD 150606|PD150606|cas 181183-52-8|DC Chemicals
PD 150606|PD150606|cas 181183-52-8|DC Chemicals
PD 150606 is a selective, cell-permeable non-peptide calpain inhibitor (Ki values for ν and m-calpains are 0.21 and 0.37 μM respectively).
Product name: PD 150606 | Cat No. DC8283 |Cas: 179528-45-1 |Other names: PD150606,PD-150606,PD 150606 |Molecule formular: C9H7IO2S |Molecule Weight: 306.12 |Purity>98%
PD 150606 is a selective, cell-permeable non-peptide calpain inhibitor (Ki values for ν and m-calpains are 0.21 and 0.37 μM respectively)
For research and scientific purpose only, not for human use.
PD 150606 is a selective, cell-permeable non-peptide calpain inhibitor (Ki values for ν and m-calpains are 0.21 and 0.37 μM respectively).
Product name: PD 150606 | Cat No. DC8283 |Cas: 179528-45-1 |Other names: PD150606,PD-150606,PD 150606 |Molecule formular: C9H7IO2S |Molecule Weight: 306.12 |Purity>98%
PD 150606 is a selective, cell-permeable non-peptide calpain inhibitor (Ki values for ν and m-calpains are 0.21 and 0.37 μM respectively)
For research and scientific purpose only, not for human use.
2015年9月15日星期二
GSK 2256294A|GSK2256294|cas 1142090-23-0|DC Chemicals
GSK 2256294A|GSK2256294|cas 1142090-23-0|DC Chemicals
GSK2256294A is a potent, reversible, tight binding inhibitor of isolated recombinant human sEH (IC50 value 27 pM), and displays potent inhibition against the rat (IC50 = 61 pM) and murine (IC50 = 189 pM) orthologs of sEH.
Product name: GSK 2256294A | Cat No. DC8282 |Cas: 1142090-23-0 |Other names: GSK 2256294,GSK-2256294,GSK2256294,GSK-2256294A,GSK2256294A |Molecule formular: C21H24F3N7O |Molecule Weight: 447.46 |Purity>98%
GSK2256294A is a potent, reversible, tight binding inhibitor of isolated recombinant human sEH (IC50 value 27 pM), and displays potent inhibition against the rat (IC50 = 61 pM) and murine (IC50 = 189 pM) orthologs of sEH.
For research and scientific purpose only, not for human use.
GSK2256294A is a potent, reversible, tight binding inhibitor of isolated recombinant human sEH (IC50 value 27 pM), and displays potent inhibition against the rat (IC50 = 61 pM) and murine (IC50 = 189 pM) orthologs of sEH.
Product name: GSK 2256294A | Cat No. DC8282 |Cas: 1142090-23-0 |Other names: GSK 2256294,GSK-2256294,GSK2256294,GSK-2256294A,GSK2256294A |Molecule formular: C21H24F3N7O |Molecule Weight: 447.46 |Purity>98%
GSK2256294A is a potent, reversible, tight binding inhibitor of isolated recombinant human sEH (IC50 value 27 pM), and displays potent inhibition against the rat (IC50 = 61 pM) and murine (IC50 = 189 pM) orthologs of sEH.
For research and scientific purpose only, not for human use.
ozanimod (RPC1063)|S1P1R modulator|DC Chemicals
ozanimod (RPC1063)|S1P1R modulator|DC Chemicals
ozanimod (RPC1063) is a selective S1P1R modulator
Product name: ozanimod (RPC1063) | Cat No. DC8281 |Cas: 1306760-87-1 |Other names: RPC1063,RPC-1063,RPC 1063 |Molecule formular: C23H24N4O3 |Molecule Weight: 404.46 |Purity>98%
ozanimod (RPC1063) is a selective S1P1R modulator
For research and scientific purpose only, not for human use.
ozanimod (RPC1063) is a selective S1P1R modulator
Product name: ozanimod (RPC1063) | Cat No. DC8281 |Cas: 1306760-87-1 |Other names: RPC1063,RPC-1063,RPC 1063 |Molecule formular: C23H24N4O3 |Molecule Weight: 404.46 |Purity>98%
ozanimod (RPC1063) is a selective S1P1R modulator
For research and scientific purpose only, not for human use.
BLU-9931,BLU9931|FGFR4 inhibitor|DC Chmeicals
BLU-9931,BLU9931|FGFR4 inhibitor|DC Chmeicals
BLU9931 is the first selective small molecule inhibitor of FGFR4 with IC50 of 3 nM; less potent for FGFR1/2/3(IC50> 150 nM).
Product name: BLU-9931 | Cat No. DC8280 |Cas: 1538604-68-0 |Other names: BLU-9931,BLU 9931,BLU9931 |Molecule formular: C26H22Cl2N4O3 |Molecule Weight: 509.38 |Purity>98%
BLU9931 is the first selective small molecule inhibitor of FGFR4 with IC50 of 3 nM; less potent for FGFR1/2/3(IC50> 150 nM).
For research and scientific purpose only, not for human use.
BLU9931 is the first selective small molecule inhibitor of FGFR4 with IC50 of 3 nM; less potent for FGFR1/2/3(IC50> 150 nM).
Product name: BLU-9931 | Cat No. DC8280 |Cas: 1538604-68-0 |Other names: BLU-9931,BLU 9931,BLU9931 |Molecule formular: C26H22Cl2N4O3 |Molecule Weight: 509.38 |Purity>98%
BLU9931 is the first selective small molecule inhibitor of FGFR4 with IC50 of 3 nM; less potent for FGFR1/2/3(IC50> 150 nM).
For research and scientific purpose only, not for human use.
SR9243|SR 9243|LXR inhibitor|DC Chemicals
SR9243|SR 9243|LXR inhibitor|DC Chemicals
SR9243 is a new inhibitor of The nuclear receptor liver-X-receptor (LXR),inducing LXR-corepressor interaction.
Product name: SR9243 | Cat No. DC8279 |Cas: 1613028-81-1 |Other names: SR 9243,SR9243,SR-9243 |Molecule formular: C31H32BrN04S2 |Molecule Weight: 626.62 |Purity>98%
SR9243 is a new inhibitor of The nuclear receptor liver-X-receptor (LXR),inducing LXR-corepressor interaction.
For research and scientific purpose only, not for human use.
SR9243 is a new inhibitor of The nuclear receptor liver-X-receptor (LXR),inducing LXR-corepressor interaction.
Product name: SR9243 | Cat No. DC8279 |Cas: 1613028-81-1 |Other names: SR 9243,SR9243,SR-9243 |Molecule formular: C31H32BrN04S2 |Molecule Weight: 626.62 |Purity>98%
SR9243 is a new inhibitor of The nuclear receptor liver-X-receptor (LXR),inducing LXR-corepressor interaction.
For research and scientific purpose only, not for human use.
BVT-14225|11b-HSD1 inhibitor|DC Chemicals
BVT-14225|11b-HSD1 inhibitor|DC Chemicals
BVT 14225 is a new selective 11b-HSD1 inhibitor, it belongs to a class of arylsulfonamidothiazoles with in vitro and in vivo antidiabetic effects
Product name: BVT-14225 | Cat No. DC8278 |Cas: 376638-65-2 |Other names: BVT14225,BVT 14225 |Molecule formular: C16H20ClN3O3S2 |Molecule Weight: 401.9 |Purity>98%
BVT 14225 is a new selective 11b-HSD1 inhibitor, it belongs to a class of arylsulfonamidothiazoles with in vitro and in vivo antidiabetic effects
For research and scientific purpose only, not for human use.
BVT 14225 is a new selective 11b-HSD1 inhibitor, it belongs to a class of arylsulfonamidothiazoles with in vitro and in vivo antidiabetic effects
Product name: BVT-14225 | Cat No. DC8278 |Cas: 376638-65-2 |Other names: BVT14225,BVT 14225 |Molecule formular: C16H20ClN3O3S2 |Molecule Weight: 401.9 |Purity>98%
BVT 14225 is a new selective 11b-HSD1 inhibitor, it belongs to a class of arylsulfonamidothiazoles with in vitro and in vivo antidiabetic effects
For research and scientific purpose only, not for human use.
E 2012|γ-secretase modulator|DC Chemicals
E 2012|γ-secretase modulator|DC Chemicals
E 2012 is a potent γ-secretase modulator.
Product name: E-2012 | Cat No. DC8277 |Cas: 870843-42-8 |Other names: E2012,E 2012,E-2012 |Molecule formular: C25H26FN3O2 |Molecule Weight: 419.49 |Purity>98%
E 2012 is a potent γ-secretase modulator
For research and scientific purpose only, not for human use.
E 2012 is a potent γ-secretase modulator.
Product name: E-2012 | Cat No. DC8277 |Cas: 870843-42-8 |Other names: E2012,E 2012,E-2012 |Molecule formular: C25H26FN3O2 |Molecule Weight: 419.49 |Purity>98%
E 2012 is a potent γ-secretase modulator
For research and scientific purpose only, not for human use.
Apilimod mesylate|STA 5326|IL-12/IL-23 inhibitor|DC Chemicals
Apilimod mesylate|STA 5326|IL-12/IL-23 inhibitor|DC Chemicals
Apilimod(STA 5326) mesylate is a potent IL-12/IL-23 inhibitor, IL-12 production in cultures of IFN-r/LPS–stimulated human PBMCs is strongly inhibited by STA-5326 with an IC50 of 10 nM.
Product name: Apilimod mesylate | Cat No. DC8276 |Cas: 870087-36-8 |Other names: STA 5326 mesylate; STA5326 mesylate; STA-5326 mesylate |Molecule formular: C25H34N6O8S2 |Molecule Weight: 610.7 |Purity>98%
Apilimod(STA 5326) mesylate is a potent IL-12/IL-23 inhibitor, IL-12 production in cultures of IFN-r/LPS–stimulated human PBMCs is strongly inhibited by STA-5326 with an IC50 of 10 nM.
For research and scientific purpose only, not for human use.
Apilimod(STA 5326) mesylate is a potent IL-12/IL-23 inhibitor, IL-12 production in cultures of IFN-r/LPS–stimulated human PBMCs is strongly inhibited by STA-5326 with an IC50 of 10 nM.
Product name: Apilimod mesylate | Cat No. DC8276 |Cas: 870087-36-8 |Other names: STA 5326 mesylate; STA5326 mesylate; STA-5326 mesylate |Molecule formular: C25H34N6O8S2 |Molecule Weight: 610.7 |Purity>98%
Apilimod(STA 5326) mesylate is a potent IL-12/IL-23 inhibitor, IL-12 production in cultures of IFN-r/LPS–stimulated human PBMCs is strongly inhibited by STA-5326 with an IC50 of 10 nM.
For research and scientific purpose only, not for human use.
Apilimod|STA 5326|IL-12/IL-23 inhibitor|DC Chemicals
Apilimod|STA 5326|IL-12/IL-23 inhibitor|DC Chemicals
Apilimod(STA 5326) is a potent IL-12/IL-23 inhibitor, IL-12 production in cultures of IFN-r/LPS–stimulated human PBMCs is strongly inhibited by STA-5326 with an IC50 of 10 nM.
Product name: Apilimod | Cat No. DC8275 |Cas: 541550-19-0 |Other names: STA 5326; STA5326; STA-5326 |Molecule formular: C23H26N6O2 |Molecule Weight: 418.49 |Purity>98%
Apilimod(STA 5326) is a potent IL-12/IL-23 inhibitor, IL-12 production in cultures of IFN-r/LPS–stimulated human PBMCs is strongly inhibited by STA-5326 with an IC50 of 10 nM.
For research and scientific purpose only, not for human use.
Apilimod(STA 5326) is a potent IL-12/IL-23 inhibitor, IL-12 production in cultures of IFN-r/LPS–stimulated human PBMCs is strongly inhibited by STA-5326 with an IC50 of 10 nM.
Product name: Apilimod | Cat No. DC8275 |Cas: 541550-19-0 |Other names: STA 5326; STA5326; STA-5326 |Molecule formular: C23H26N6O2 |Molecule Weight: 418.49 |Purity>98%
Apilimod(STA 5326) is a potent IL-12/IL-23 inhibitor, IL-12 production in cultures of IFN-r/LPS–stimulated human PBMCs is strongly inhibited by STA-5326 with an IC50 of 10 nM.
For research and scientific purpose only, not for human use.
Dihydroethidium|superoxide indicator|DC Chemicals
Dihydroethidium|superoxide indicator|DC Chemicals
Dihydroethidium(Hydroethidine; PD-MY 003) is a superoxide indicator; exhibits blue-fluorescence in the cytosol until oxidized, where it intercalates within the cell's DNA, staining its nucleus a bright fluorescent red.
Product name: Dihydroethidium | Cat No. DC8274 |Cas: 104821-25-2 |Other names: Hydroethidine; PD-MY 003 |Molecule formular: C21H21N3 |Molecule Weight: 315.41 |Purity>98%
Dihydroethidium(Hydroethidine; PD-MY 003) is a superoxide indicator; exhibits blue-fluorescence in the cytosol until oxidized, where it intercalates within the cell's DNA, staining its nucleus a bright fluorescent red.
For research and scientific purpose only, not for human use.
Dihydroethidium(Hydroethidine; PD-MY 003) is a superoxide indicator; exhibits blue-fluorescence in the cytosol until oxidized, where it intercalates within the cell's DNA, staining its nucleus a bright fluorescent red.
Product name: Dihydroethidium | Cat No. DC8274 |Cas: 104821-25-2 |Other names: Hydroethidine; PD-MY 003 |Molecule formular: C21H21N3 |Molecule Weight: 315.41 |Purity>98%
Dihydroethidium(Hydroethidine; PD-MY 003) is a superoxide indicator; exhibits blue-fluorescence in the cytosol until oxidized, where it intercalates within the cell's DNA, staining its nucleus a bright fluorescent red.
For research and scientific purpose only, not for human use.
OAC-2|IPCS reprogramming enhancer|DC Chemicals
OAC-2|IPCS reprogramming enhancer|DC Chemicals
OAC2 is an Oct4-activating compound which activates expression through the Oct4 gene promoter; enhances reprogramming efficiency by increasing the rate of production of induced pluripotent stem cells (iPSCs) from embryonic fibroblasts; an analog of OAC1.
Product name: OAC2 | Cat No. DC8273 |Cas: 6019-39-2 |Other names: OAC-2,OAC 2 |Molecule formular: C15H12N2O |Molecule Weight: 236.27 |Purity>98%
OAC2 is an Oct4-activating compound which activates expression through the Oct4 gene promoter; enhances reprogramming efficiency by increasing the rate of production of induced pluripotent stem cells (iPSCs) from embryonic fibroblasts; an analog of OAC1.
For research and scientific purpose only, not for human use.
OAC2 is an Oct4-activating compound which activates expression through the Oct4 gene promoter; enhances reprogramming efficiency by increasing the rate of production of induced pluripotent stem cells (iPSCs) from embryonic fibroblasts; an analog of OAC1.
Product name: OAC2 | Cat No. DC8273 |Cas: 6019-39-2 |Other names: OAC-2,OAC 2 |Molecule formular: C15H12N2O |Molecule Weight: 236.27 |Purity>98%
OAC2 is an Oct4-activating compound which activates expression through the Oct4 gene promoter; enhances reprogramming efficiency by increasing the rate of production of induced pluripotent stem cells (iPSCs) from embryonic fibroblasts; an analog of OAC1.
For research and scientific purpose only, not for human use.
U-104|carbonic anhydrase(CA) inhibitor|DC Chemicals
U-104|carbonic anhydrase(CA) inhibitor|DC Chemicals
U-104 is a potent carbonic anhydrase (CA) inhibitor for CA IX and CA XII with Ki of 45.1 nM and 4.5 nM; low inhibition for CA I and CA II.
Product name: U-104 | Cat No. DC8272 |Cas: 178606-66-1 |Other names: NSC-213841; MST-104，U104，U 104 |Molecule formular: C13H12FN3O3S |Molecule Weight: 309.32 |Purity>98%
U-104 is a potent carbonic anhydrase (CA) inhibitor for CA IX and CA XII with Ki of 45.1 nM and 4.5 nM; low inhibition for CA I and CA II.
For research and scientific purpose only, not for human use.
U-104 is a potent carbonic anhydrase (CA) inhibitor for CA IX and CA XII with Ki of 45.1 nM and 4.5 nM; low inhibition for CA I and CA II.
Product name: U-104 | Cat No. DC8272 |Cas: 178606-66-1 |Other names: NSC-213841; MST-104，U104，U 104 |Molecule formular: C13H12FN3O3S |Molecule Weight: 309.32 |Purity>98%
U-104 is a potent carbonic anhydrase (CA) inhibitor for CA IX and CA XII with Ki of 45.1 nM and 4.5 nM; low inhibition for CA I and CA II.
For research and scientific purpose only, not for human use.
NSC41589|NSC-41589|DC Chemicals
NSC41589|NSC-41589|DC Chemicals
N-[2-(methylsulfanyl) phenyl]acetamide.
Product name: NSC-41589 | Cat No. DC8271 |Cas: 6310-41-4 |Other names: NSC41589; NSC 41589 |Molecule formular: C9H11NOS |Molecule Weight: 181.25 |Purity>98%
N-[2-(methylsulfanyl) phenyl]acetamide.
For research and scientific purpose only, not for human use.
N-[2-(methylsulfanyl) phenyl]acetamide.
Product name: NSC-41589 | Cat No. DC8271 |Cas: 6310-41-4 |Other names: NSC41589; NSC 41589 |Molecule formular: C9H11NOS |Molecule Weight: 181.25 |Purity>98%
N-[2-(methylsulfanyl) phenyl]acetamide.
For research and scientific purpose only, not for human use.
BML277|Chk2 Inhibitor II|DC Chemicals
BML277|Chk2 Inhibitor II|DC Chemicals
BML-277 (C 3742) is a selective Chk2 (checkpoint kinase 2) inhibitor with an IC50 of 15 nM.
Product name: BML-277 | Cat No. DC8270 |Cas: 516480-79-8 |Other names: Chk2 Inhibitor II; C 3742; BML277; BML 277 |Molecule formular: C20H14ClN3O2 |Molecule Weight: 363.8 |Purity>98%
BML-277 (C 3742) is a selective Chk2 (checkpoint kinase 2) inhibitor with an IC50 of 15 nM.
For research and scientific purpose only, not for human use.
BML-277 (C 3742) is a selective Chk2 (checkpoint kinase 2) inhibitor with an IC50 of 15 nM.
Product name: BML-277 | Cat No. DC8270 |Cas: 516480-79-8 |Other names: Chk2 Inhibitor II; C 3742; BML277; BML 277 |Molecule formular: C20H14ClN3O2 |Molecule Weight: 363.8 |Purity>98%
BML-277 (C 3742) is a selective Chk2 (checkpoint kinase 2) inhibitor with an IC50 of 15 nM.
For research and scientific purpose only, not for human use.
NS6180|Ca2+-activated K+ channel (KCa3.1) inhibitor|DC Chemicals
NS6180|Ca2+-activated K+ channel (KCa3.1) inhibitor|DC Chemicals
NS6180 is a novel inhibitor of the intermediate-conductance Ca2+-activated K+ channel (KCa3.1)
Product name: NS6180 | Cat No. DC8269 |Cas: 353262-04-1 |Other names: NS6180,NS-6180，NS 6180 |Molecule formular: C16H12F3NOS |Molecule Weight: 323.33 |Purity>98%
NS6180 is a novel inhibitor of the intermediate-conductance Ca2+-activated K+ channel (KCa3.1)
For research and scientific purpose only, not for human use.
NS6180 is a novel inhibitor of the intermediate-conductance Ca2+-activated K+ channel (KCa3.1)
Product name: NS6180 | Cat No. DC8269 |Cas: 353262-04-1 |Other names: NS6180,NS-6180，NS 6180 |Molecule formular: C16H12F3NOS |Molecule Weight: 323.33 |Purity>98%
NS6180 is a novel inhibitor of the intermediate-conductance Ca2+-activated K+ channel (KCa3.1)
For research and scientific purpose only, not for human use.
Eliprodil|NMDA receptor inhibitor|DC Chemicals
Eliprodil|NMDA receptor inhibitor|DC Chemicals
Eliprodil is a non-competitive NMDA receptor antagonist that acts at the polyamine modulatory site.
Product name: Eliprodil | Cat No. DC8268 |Cas: 119431-25-3 |Other names: |Molecule formular: C20H23ClFNO |Molecule Weight: 347.86 |Purity>98%
Eliprodil is a non-competitive NMDA receptor antagonist that acts at the polyamine modulatory site.
For research and scientific purpose only, not for human use.
Eliprodil is a non-competitive NMDA receptor antagonist that acts at the polyamine modulatory site.
Product name: Eliprodil | Cat No. DC8268 |Cas: 119431-25-3 |Other names: |Molecule formular: C20H23ClFNO |Molecule Weight: 347.86 |Purity>98%
Eliprodil is a non-competitive NMDA receptor antagonist that acts at the polyamine modulatory site.
For research and scientific purpose only, not for human use.
SW033291|SW-033291|15-PGDH enzyme inhibitor|DC Chemicals
SW033291|SW-033291|15-PGDH enzyme inhibitor|DC Chemicals
SW033291 is a potent inhibitor of 15-PGDH enzyme with IC50 value of 1.5 nM and dissociation constant Ki app value of 0.1 nM.
Product name: SW033291 | Cat No. DC8267 |Cas: 459147-39-8 |Other names: SW033291,SW-033291,SW033291,SW 033291 |Molecule formular: C21H22N2OS3 |Molecule Weight: 414.61 |Purity>98%
SW033291 is a potent inhibitor of 15-PGDH enzyme with IC50 value of 1.5 nM and dissociation constant Ki app value of 0.1 nM.
For research and scientific purpose only, not for human use.
SW033291 is a potent inhibitor of 15-PGDH enzyme with IC50 value of 1.5 nM and dissociation constant Ki app value of 0.1 nM.
Product name: SW033291 | Cat No. DC8267 |Cas: 459147-39-8 |Other names: SW033291,SW-033291,SW033291,SW 033291 |Molecule formular: C21H22N2OS3 |Molecule Weight: 414.61 |Purity>98%
SW033291 is a potent inhibitor of 15-PGDH enzyme with IC50 value of 1.5 nM and dissociation constant Ki app value of 0.1 nM.
For research and scientific purpose only, not for human use.
GW 627368X|EP4 receptor inhibitor|DC Chemicals
GW 627368X|EP4 receptor inhibitor|DC Chemicals
GW 627368X is a selective prostanoid EP4 receptor competitive antagonist with additional affinity at TP receptors (pKi values are 7.0 and 6.8 in competition radioligand bioassays).
Product name: GW-627368X | Cat No. DC8266 |Cas: 439288-66-1 |Other names: GW 627368,GW-627368,GW627368,GW-627368X,GW627368X，GW 627368X |Molecule formular: C30H28N2O6S |Molecule Weight: 544.62 |Purity>98%
GW 627368X is a selective prostanoid EP4 receptor competitive antagonist with additional affinity at TP receptors (pKi values are 7.0 and 6.8 in competition radioligand bioassays).
For research and scientific purpose only, not for human use.
GW 627368X is a selective prostanoid EP4 receptor competitive antagonist with additional affinity at TP receptors (pKi values are 7.0 and 6.8 in competition radioligand bioassays).
Product name: GW-627368X | Cat No. DC8266 |Cas: 439288-66-1 |Other names: GW 627368,GW-627368,GW627368,GW-627368X,GW627368X，GW 627368X |Molecule formular: C30H28N2O6S |Molecule Weight: 544.62 |Purity>98%
GW 627368X is a selective prostanoid EP4 receptor competitive antagonist with additional affinity at TP receptors (pKi values are 7.0 and 6.8 in competition radioligand bioassays).
For research and scientific purpose only, not for human use.
Endoxifen|tamoxifen metabolite|DC Chemicals
Endoxifen|tamoxifen metabolite|DC Chemicals
Endoxifen is a Estrogen receptor α (ERα) ligand; potent antiestrogen,an active metabolite of the cancer drug tamoxifen.
Product name: Endoxifen | Cat No. DC8265 |Cas: 110025-28-0 |Other names: N/A |Molecule formular: C25H27NO2 |Molecule Weight: 373.49 |Purity>98%
Endoxifen is a Estrogen receptor α (ERα) ligand; potent antiestrogen,an active metabolite of the cancer drug tamoxifen.
For research and scientific purpose only, not for human use.
Endoxifen is a Estrogen receptor α (ERα) ligand; potent antiestrogen,an active metabolite of the cancer drug tamoxifen.
Product name: Endoxifen | Cat No. DC8265 |Cas: 110025-28-0 |Other names: N/A |Molecule formular: C25H27NO2 |Molecule Weight: 373.49 |Purity>98%
Endoxifen is a Estrogen receptor α (ERα) ligand; potent antiestrogen,an active metabolite of the cancer drug tamoxifen.
For research and scientific purpose only, not for human use.
MM41|MM-41|Bcl-2/K-Ras inhibitor|DC Chemicals
MM41|MM-41|Bcl-2/K-Ras inhibitor|DC Chemicals
MM41 is a quadruplex-interactive compound which binds strongly to the quadruplexes encoded in the promoter sequences of the BCL-2 and k-RAS genes.
Product name: MM-41 | Cat No. DC8264 |Cas: N/A |Other names: MM41,MM 41 |Molecule formular: C44H66NO6 |Molecule Weight: 830.52 |Purity>98%
MM41 is a quadruplex-interactive compound which binds strongly to the quadruplexes encoded in the promoter sequences of the BCL-2 and k-RAS genes.
For research and scientific purpose only, not for human use.
MM41 is a quadruplex-interactive compound which binds strongly to the quadruplexes encoded in the promoter sequences of the BCL-2 and k-RAS genes.
Product name: MM-41 | Cat No. DC8264 |Cas: N/A |Other names: MM41,MM 41 |Molecule formular: C44H66NO6 |Molecule Weight: 830.52 |Purity>98%
MM41 is a quadruplex-interactive compound which binds strongly to the quadruplexes encoded in the promoter sequences of the BCL-2 and k-RAS genes.
For research and scientific purpose only, not for human use.
Bikinin|Glycogen synthase kinase inhibitor|DC Chemicals
Bikinin|Glycogen synthase kinase inhibitor|DC Chemicals
Bikinin is a strong activator of brassinosteroid (BR) signaling.
Product name: Bikinin | Cat No. DC8263 |Cas: 188011-69-0 |Other names: |Molecule formular: C9H9BrN2O3 |Molecule Weight: 273.08 |Purity>98%
Bikinin is a strong activator of brassinosteroid (BR) signaling.
Bikinin is a strong activator of brassinosteroid (BR) signaling.
Product name: Bikinin | Cat No. DC8263 |Cas: 188011-69-0 |Other names: |Molecule formular: C9H9BrN2O3 |Molecule Weight: 273.08 |Purity>98%
Bikinin is a strong activator of brassinosteroid (BR) signaling.
For research and scientific purpose only, not for human use.
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