URB754(URB-754)|MAGL inhibitor|DC Chemicals
URB754 is reported to be a potent, noncompetitive inhibitor of monoacylglycerol lipase (MAGL), exhibiting an IC50 of 200 nM for the recombinant rat brain enzyme.
Product name: URB754 |Cat No. DC8130|Other names: URB754,URB 754,URB-754|Cas: 86672-58-4|Molecule Weight: 266.29|Molecule Formular: C16H14N2O2| Purity: >98%
URB-754 is a new class of designer drug and 12 synthetic cannabinoids detected in illegal products.URB-754 was reported to inhibit an endocannabinoid deactivating enzyme.Subsequent studies have shown that that URB-754 does not inhibit recombinant MAG Lipase and that the original activity was due to a contaminant, bis(methylthio)mercurane, in another commercial source. URB-754 is an inhibitor of FAAH.
For research and scientific purpose only, not for human use.
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