Tosedostat (CHR2797)|aminopeptidase inhibitor|DC Chemicals

Tosedostat (CHR2797)|aminopeptidase inhibitor|DC Chemicals
CHR-2797 is an aminopeptidase inhibitor, with IC50 values of 100 nM for LAP3 (LAP), 150 nM for PSAP (PuSA) and 220 nM for CD13 (Aminopeptidase N).

Catlog: DC8116| Product name: Tosedostat (CHR2797)| Cas: 238750-77-1| Other names: CHR 2797,CHR-2797| Molecule Formula: C21H30N2O6| MW: 406.47. Purity: >98%

Price: 100mg: 500 USD; 250mg: 900 USD; 1000mg: 1900 USD

CHR-2797 is an aminopeptidase inhibitor, with IC50 values of 100 nM for LAP3 (LAP), 150 nM for PSAP (PuSA) and 220 nM for CD13 (Aminopeptidase N). CHR-2797 is converted in cells to the active acid metabolite, CHR-79888, which is a significant inhibitor of Leukotriene A4 hydrolase with an IC50 of 8 nM. CHR-2797 exhibits profound anti-proliferative effects against a range of cancer cell lines such as U-937, HL-60, KG-1 and GDM-1.

For research and scientific purpose only, not for human use.