I-BRD9|cas 1182367-47-0|DC Chemicals

I-BRD9|cas 1182367-47-0|DC Chemicals

I-BRD9 is a potent and selective BRD9 inhibitor (pIC50 = 7.3). Exhibits >70-fold selectivity for BRD9 over a panel of 34 other bromodomains and >700-fold selectivity over the BET family.

Product Name: I-BRD9|Cat No: DC9658|Cas: 1714146-59-4|Molecule Formular: C22H22F3N3O3S2|Molecule Weight: 497.55|Other names: I-BRD9

I-BRD9 is a potent and selective binder to BRD9 with a pIC50 in a Time-Resolved FRET assay of 7.3. BRD4 was used as a representative member of the BET family for initial selectivity screening, I-BRD9 displayed a pIC50 of 5.3 against this protein. I-BRD9 binds to endogenous BRD9 in a chemoproteomic assay and shows good selectivity over the BET family member BRD3.

For research only, not for human use.