2014年8月11日星期一

VX-11e|cas 896720-20-0| DC Chem|Supplier|Price|Buy  

VX-11e|cas 896720-20-0| DC Chem|Supplier|Price|Buy
DC Chemicals Supply: VX-11e|cas 896720-20-0,Purity: >98% ,Cat No. DC7242, In stock.

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VX-11e|cas 896720-20-0 ,Synonym: VX 11e  ,Chemical name: 4-[2-(2-chloro-4-fluoroanilino)-5-methylpyrimidin-4-yl]-N-[(1S)-1-(3-chlorophenyl)-2-hydroxyethyl]-1H-pyrrole-2-carboxamide ,Molecular Formula: 896720-20-0, pyrimidylpyrrole, 11e, CHEMBL583042, CS-0995, NCGC00242487-01, HY-14178, KB-81470, VX-11e|896720-20-0 ,MW:500.352303

VX-11e, cas 896720-20-0,Purity: >98%, Best Price and quality from DC Chemicals. VX-11e is a potent, selective, and orally bioavailable inhibitor of ERK (Extracellular Signal-Regulated Kinase); antitumor agent.

Potent and selective extracellular signal-related kinase 2 (ERK2) inhibitor (Ki values are <2, 395, 540 and 852 nM for ERK2, GSK-3, Aurora Kinase A and Cdk2 respectively). Potently blocks proliferation of HT29 cells (IC50 = 48 nM). Orally bioavailable.

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