2014年8月30日星期六

lexibulin (CYT997) supplier|cas 917111-44-5 |DC Chemicals|Supplier|Price|Buy  

lexibulin (CYT997) supplier|cas 917111-44-5 |DC Chemicals|Supplier|Price|Buy

DC Chemicals Supply: lexibulin (CYT997) supplier,cas 917111-44-5, Cat No. DC5134, In stock

Contact: website: www.dcchemicals.com,
sales@dcchemicals.com,order@dcchemicals.com,info@dcchemicals.com,
Tel: +86-21-61454686;Fax:+86-21-61642863;

Product name: lexibulin (CYT997), Synonym: CYT997; CYT-997; CYT 997. lexibulin., Cat No. DC5134, Cas: 917111-44-5, Chemical Name:N-Ethyl-N'-[2-methoxy-4-[5-methyl-4-[[(1S)-1-(3-pyridinyl)butyl]amino]-2-pyrimidinyl]phenyl]urea, Molecular Formula: C24H30N6O2, MW: 434.534

lexibulin (CYT997),cas 917111-44-5, Purity: >98%. Best Price and quality in the market,DC Chemicals,Primary Manufacturer, confirmed by HNMR and HPLC. CYT997 is a potent microtubule polymerization inhibitor with IC50 of 10-100 nM in cancer cell lines. Phase 1/2.

lexibulin, also known as CYT997,  is an orally bioavailable small-molecule with tubulin-inhibiting, vascular-disrupting, and potential antineoplastic activities. Lexibulin inhibits tubulin polymerization in tumor blood vessel endothelial cells and tumor cells, blocking the formation of the mitotic spindle and leading to cell cycle arrest at the G2/M phase; this may result in disruption of the tumor vasculature and tumor blood flow, and tumor cell death.

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