GSK269962A(GSK269962) |cas 850664-21-0| DC Chem|Supplier|Price|Buy
GSK269962A(GSK269962) |cas 850664-21-0| DC Chem|Supplier|Price|Buy
DC Chemicals Supply: GSK269962A(GSK269962) |cas 850664-21-0,Purity: >98% ,Cat No. DC7249, In stock.
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GSK269962A(GSK269962) |cas 850664-21-0 ,Synonym: GSK 269962A; GSK-269962A; GSK269962; GSK 269962; GSK-269962 ,Chemical name: N-[3-[[2-(4-Amino-1,2,5-oxadiazol-3-yl)-1-ethyl-1H-imidazo[4,5-c]pyridin-6-yl]oxy]phenyl]-4-[2-(4-morpholinyl)ethoxy]benzamide ,Molecular Formula: C29H30N8O5 ,MW:570.6
GSK269962A(GSK269962) , cas 850664-21-0,Purity: >98%, Best Price and quality from DC Chemicals. GSK269962A(GSK269962) is a potent ROCK inhibitor (IC50 values are 1.6 and 4 nM for recombinant human ROCK1 and ROCK2 respectively); displays greater than 30-fold selectivity for ROCK against a panel of serine/threonine kinases.
Potent Rho kinase (ROCK) inhibitor (IC50 values are 1.6 and 4 nM for recombinant human ROCK1 and ROCK2 respectively). Displays greater than 30-fold selectivity for ROCK against a panel of serine/threonine kinases. Induces vasorelaxation in preconstricted rat aorta (IC50 = 35 nM); lowers blood pressure in a rat model of hypertension.
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