2014年8月10日星期日

SB-657510|cas 474960-44-6| DC Chem|Supplier|Price|Buy  

SB-657510|cas 474960-44-6| DC Chem|Supplier|Price|Buy
DC Chemicals Supply: SB-657510|cas 474960-44-6,Purity: >98% ,Cat No. DC7288, In stock.

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SB-657510|cas 474960-44-6 ,Synonym:  ,Chemical name: 2-Bromo-N-[4-chloro-3-[[(3R)-1-methyl-3-pyrrolidinyl]oxy]phenyl]-4,5-dimethoxybenzenesulfonamide ,Molecular Formula: C19H22BrClN2O5S ,MW:505.81

SB-657510, cas 474960-44-6,Purity: >98%, Best Price and quality from DC Chemicals. Selective urotensin-II (UT) receptor antagonist (Ki values are 61, 17, 30, 65 and 56 nM at human, monkey, cat, rat and mouse receptors respectively). Inhibits U-II-induced intracellular Ca2+ mobilization (IC50 = 180 nM) and antagonizes the contractile action of U-II in isolated mammalian arteries and aortae (EC50 = 50 - 189 nM).

Selective urotensin-II (UT) receptor antagonist (Ki values are 61, 17, 30, 65 and 56 nM at human, monkey, cat, rat and mouse receptors respectively). Inhibits U-II-induced intracellular Ca2+mobilization (IC50 = 180 nM) and antagonizes the contractile action of U-II in isolated mammalian arteries and aortae (EC50 = 50 - 189 nM).

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