2016年1月7日星期四

SB-399885|5-HT6 antagonist|DC Chemicals

SB-399885|5-HT6 antagonist|DC Chemicals

Potent, brain penetrant, orally active 5-HT6 antagonist. Displays > 200-fold selectivity for 5-HT6 over other 5-HT receptors (pKi values are 9.11, 8.81 and 9.02  for human recombinant, native rat and native human 5-HT6 receptors respectively).

Product Name: SB-399885 HCl |Catalog Number: DC8483 |CAS 402713-80-8  |Other names: SB-399885,SB 399885,SB399885 |Chemical Name: N-(3,5-Dichloro-2-methoxyphenyl)-4-methoxy-3-(1-piperazinyl)benzenesulfonamide hydrochloride |Molecule Formular: C18H21Cl2N3O4S.HCl |MW: 482.81

Potent, brain penetrant, orally active 5-HT6 antagonist. Displays > 200-fold selectivity for 5-HT6 over other 5-HT receptors (pKi values are 9.11, 8.81 and 9.02  for human recombinant, native rat and native human 5-HT6 receptors respectively).

For research and scientific purpose only, not for human use.

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