CB1-IN-1 is a peripherally restricted CB1R antagonist, with Ki of 0.3 nM and 21 nM for CB1R (EC50 = 3 nM) and CB2R, respectively.
Product Name: CB1-IN-1 |Catalog Number: DC8719 |CAS 1429239-98-4 |Other names: |Chemical Name: |Molecule Formular: C33H31Cl2F3N6O3S2 |MW: 751.67
CB1-IN-1 is a peripherally restricted CB1R antagonist, with Ki of 0.3 nM and 21 nM for CB1R (EC50 = 3 nM) and CB2R, respectively.in vivo: CB1-IN-1 is a novel peripherally restricted cannabinoid 1 receptor antagonist with significant weight-loss efficacy in diet-induced obese mice. CB1-IN-1 has great potential to ameliorate this related metabolic syndrome.
For research and scientific purpose only, not for human use!
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