GSK9311|GSK-9311|BRPF bromodomain inhibitor

GSK9311|GSK-9311|BRPF bromodomain inhibitor

GSK9311 is a potent and highly selective inhibitor of the BRPF bromodomain (BRPDF1 pIC50 = 6.0; BRPDF2 pIC50 = 4.3).

Product Name: GSK9311|Cat No: DC9907|cas: 1923851-49-3|Other Names: GSK 9311,GSK-9311

GSK9311 is a potent and highly selective inhibitor of the BRPF bromodomain (BRPDF1 pIC50 = 6.0; BRPDF2 pIC50 = 4.3). The BRPF (Bromodomain and PHD Fingercontaining) protein family are important scaffolding proteins for assembly of MYST histone acetyltransferase complexes. BRPF1 (bromodomain and PHD finger containing protein 1) is involved in the epigenetic regulation of gene expression and have been implicated in human cancer.

For the research and scientific use only, not for human use!