Acumapimod |cas 836683-15-9

Acumapimod |cas 836683-15-9

DC Chemicals, Website: www.dcchemicals.com

Product Name: Acumapimod|Cas Number: 836683-15-9| Catalog Number: DC10417

Acumapimod (BCT197) is an orally active p38 MAP kinase inhibitor, with an IC50 of less than 1 μM for p38α.

Acumapimod is an inhibitor of p38α with an IC50 value of less than 1 μM.BCT197 is an oral low-molecular-weight p38 inhibitor currently in development for the treatment of several inflammatory conditions, including chronic obstructive pulmonary disease (COPD). Intermittent short-term dosing of BCT197 (75 mg on days 1 and 6) shows a marked improvement in lung function in COPD patients[2].