CPI-169 (R) supplier|CPI169|DC Chemicals

CPI-169 (R) supplier|CPI169|DC Chemicals
DC Chemicals provides CPI-169 (R), other names: CPI 169,CPI169, cas: . In stock.

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CPI-169 R is a novel and potent EZH2 inhibitor with IC50 <1 nM(inhibition of the catalytic activity of PRC2.

CPI-169 (R), other names: CPI 169,CPI169, cas: , Molecule formular: C27H36N4O5S, Molecule Weight: 528.66, Chemical name:

CPI-169, a representative compound from that effort, inhibits the catalytic activity of PRC2 with an IC50 of < 1nM, decreases cellular levels of H3K27me3 with an EC50 of 70 nM, and triggers cell cycle arrest and apoptosis in a variety of cell lines. Importantly, compound treatment triggers a sequence of downstream functional consequences of EZH2 inhibition whereby apoptosis is not induced before ten days of continuous target engagement For the detailed information of CPI-169 (R), the solubility of CPI-169 (R) in water, the solubility of CPI-169 (R) in DMSO, the solubility of CPI-169 (R) in PBS buffer, the animal experiment (test) of  CPI-169 (R), the cell expriment (test) of CPI-169 (R), the in vivo, in vitro and clinical trial test of CPI-169 (R), the EC50, IC50,and affinity,of CPI-169 (R), Please contact DC Chemicals.