2015年6月1日星期一

URB754(URB-754)|MAGL inhibitor|DC Chemicals

URB754(URB-754)|MAGL inhibitor|DC Chemicals
URB754 is reported to be a potent, noncompetitive inhibitor of monoacylglycerol lipase (MAGL), exhibiting an IC50 of 200 nM for the recombinant rat brain enzyme.

Catlog: DC8130| Product name: URB754| Cas: 86672-58-4| Other names: URB754,URB 754,URB-754| Molecule Formula: C16H14N2O2| MW: 266.29. Purity: >98%

Price: 100mg: 350 USD; 250mg: 600 USD; 1000mg: 1200 USD

URB-754 is a new class of designer drug and 12 synthetic cannabinoids detected in illegal products.URB-754 was reported to inhibit an endocannabinoid deactivating enzyme.Subsequent studies have shown that that URB-754 does not inhibit recombinant MAG Lipase and that the original activity was due to a contaminant, bis(methylthio)mercurane, in another commercial source. URB-754 is an inhibitor of FAAH.

For research and scientific purpose only, not for human use.

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