LY2119620|cas 886047-22-9|DC Chemicals

LY2119620|cas 886047-22-9|DC Chemicals

LY2119620 is a specific, and allosteric agonist of human M2 and M4 muscarinic acetylcholine receptors.

Product Name: LY2119620 |Catalog Number: DC8435 |CAS 886047-22-9 |Other names: LY2119620,LY-2119620,LY 2119620 |Chemical Name: 3-amino-5-chloro-N-cyclopropyl-4-methyl-6-[2-(4-methyl-1-piperazinyl)-2-oxoethoxy]-thieno[2,3-b]pyridine-2-carboxamide |Molecule Formular: C19H24ClN5O3S |MW: 437.94

LY2119620 displays modest allosteric agonism and positively modulates the functional G protein–signaling ability of an agonist at the M2/M4 receptor subtypes by placing the M2 and M4 receptors into an active G protein–bound state. LY2119620 enhances the potency of three muscarinic acetylcholine receptor agonists, ACh, Oxo-M and iperoxo. [1] [3H]LY2119620 can be used as a probe for the human M(2) and M(4) muscarinic receptor allosteric binding sites. [2] For the detailed information of LY2119620, the solubility of LY2119620 in water, the solubility of LY2119620 in DMSO, the solubility of LY2119620 in PBS buffer, the animal experiment (test) of  LY2119620, the cell expriment (test) of LY2119620, the in vivo, in vitro and clinical trial test of LY2119620, the EC50, IC50,and affinity,of LY2119620, For the detailed information of LY2119620, the solubility of LY2119620 in water, the solubility of LY2119620 in DMSO, the solubility of LY2119620 in PBS buffer, the animal experiment (test) of  LY2119620, the cell expriment (test) of LY2119620, the in vivo, in vitro and clinical trial test of LY2119620, the EC50, IC50,and affinity,of LY2119620, Please contact DC Chemicals.

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